1. 2-Oxoglutarate regulates binding of hydroxylated hypoxia-inducible factor to prolyl hydroxylase domain 2. Issue 25 (9th March 2018) Authors: Abboud, Martine I.; McAllister, Tom E.; Leung, Ivanhoe K. H.; Chowdhury, Rasheduzzaman; Jorgensen, Christian; Domene, Carmen; Mecinović, Jasmin; Lippl, Kerstin; Hancock, Rebecca L.; Hopkinson, Richard J.; Kawamura, Akane; Claridge, Timothy D. W.; Schofield, Christopher J. Journal: Chemical communications Issue: Volume 54:Issue 25(2018) Page Start: 3130 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. A Cell‐Permeable Ester Derivative of the JmjC Histone Demethylase Inhibitor IOX1. Issue 3 (6th February 2014) Authors: Schiller, Rachel; Scozzafava, Giuseppe; Tumber, Anthony; Wickens, James R.; Bush, Jacob T.; Rai, Ganesha; Lejeune, Clarisse; Choi, Hwanho; Yeh, Tzu‐Lan; Chan, Mun Chiang; Mott, Bryan T.; McCullagh, James S. O.; Maloney, David J.; Schofield, Christopher J.; Kawamura, Akane Journal: ChemMedChem Issue: Volume 9:Issue 3(2014:Mar.) Page Start: 566 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. An integrated platform approach enables discovery of potent, selective and ligand-competitive cyclic peptides targeting the GIP receptor. Issue 11 (2nd March 2022) Authors: Bhushan, Bhaskar; Granata, Daniele; Kaas, Christian S.; Kasimova, Marina A.; Ren, Qiansheng; Cramer, Christian N.; White, Mark D.; Hansen, Ann Maria K.; Fledelius, Christian; Invernizzi, Gaetano; Deibler, Kristine; Coleman, Oliver D.; Zhao, Xin; Qu, Xinping; Liu, Haimo; Zurmühl, Silvana S.; Kodra... Journal: Chemical science Issue: Volume 13:Issue 11(2022) Page Start: 3256 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Corrigendum to "Structure-activity studies of a macrocyclic peptide inhibitor of histone lysine demethylase 4A" [Bioorg. Med. Chem. 26/6 (2018) 1225–1231]. Issue 3 (1st February 2019) Authors: Passioura, Toby; Bhushan, Bhaskar; Tumber, Anthony; Kawamura, Akane; Suga, Hiroaki Journal: Bioorganic & medicinal chemistry Issue: Volume 27:Issue 3(2019) Page Start: 578 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Design, Synthesis and Characterization of Covalent KDM5 Inhibitors. (7th December 2018) Authors: Vazquez‐Rodriguez, Saleta; Wright, Miranda; Rogers, Catherine M.; Cribbs, Adam P.; Velupillai, Srikannathasan; Philpott, Martin; Lee, Henry; Dunford, James E.; Huber, Kilian V. M.; Robers, Matthew B.; Vasta, James D.; Thezenas, Marie‐Laetitia; Bonham, Sarah; Kessler, Benedikt; Bennett, James; Fed... Journal: Angewandte Chemie Issue: Volume 131:Number 2(2019) Page Start: 525 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Design, Synthesis and Characterization of Covalent KDM5 Inhibitors. Issue 2 (7th December 2018) Authors: Vazquez‐Rodriguez, Saleta; Wright, Miranda; Rogers, Catherine M.; Cribbs, Adam P.; Velupillai, Srikannathasan; Philpott, Martin; Lee, Henry; Dunford, James E.; Huber, Kilian V. M.; Robers, Matthew B.; Vasta, James D.; Thezenas, Marie‐Laetitia; Bonham, Sarah; Kessler, Benedikt; Bennett, James; Fed... Journal: Angewandte Chemie international edition Issue: Volume 58:Issue 2(2019) Page Start: 515 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Discovery of a Highly Selective Cell‐Active Inhibitor of the Histone Lysine Demethylases KDM2/7. (7th November 2017) Authors: Gerken, Philip A.; Wolstenhulme, Jamie R.; Tumber, Anthony; Hatch, Stephanie B.; Zhang, Yijia; Müller, Susanne; Chandler, Shane A.; Mair, Barbara; Li, Fengling; Nijman, Sebastian M. B.; Konietzny, Rebecca; Szommer, Tamas; Yapp, Clarence; Fedorov, Oleg; Benesch, Justin L. P.; Vedadi, Masoud; Kessl... Journal: Angewandte Chemie Issue: Volume 129:Number 49(2017) Page Start: 15761 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Discovery of a Highly Selective Cell‐Active Inhibitor of the Histone Lysine Demethylases KDM2/7. Issue 49 (7th November 2017) Authors: Gerken, Philip A.; Wolstenhulme, Jamie R.; Tumber, Anthony; Hatch, Stephanie B.; Zhang, Yijia; Müller, Susanne; Chandler, Shane A.; Mair, Barbara; Li, Fengling; Nijman, Sebastian M. B.; Konietzny, Rebecca; Szommer, Tamas; Yapp, Clarence; Fedorov, Oleg; Benesch, Justin L. P.; Vedadi, Masoud; Kessl... Journal: Angewandte Chemie international edition Issue: Volume 56:Issue 49(2017) Page Start: 15555 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Editorial overview: Epigenetics equals chemical biology. (August 2020) Authors: Kawamura, Akane; Ganesan, A. Journal: Current opinion in chemical biology Issue: Volume 57(2020) Page Start: A1 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. Epigenetic regulation by histone demethylases in hypoxia. (August 2015) Authors: Hancock, Rebecca L; Dunne, Kate; Walport, Louise J; Flashman, Emily; Kawamura, Akane Journal: Epigenomics Issue: Volume 7:Number 5(2015) Page Start: 791 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗