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Author/Creator Cabalu, Tamara D.

1. Cover Picture: Discovery of 5′′‐Chloro‐N‐[(5, 6‐dimethoxypyridin‐2‐yl)methyl]‐2, 2′:5′, 3′′‐terpyridine‐3′‐carboxamide (MK‐1064): A Selective Orexin 2 Receptor Antagonist (2‐SORA) for the Treatment of Insomnia (ChemMedChem 2/2014). Issue 2 (February 2014)

Authors:
Roecker, Anthony J.; Mercer, Swati P.; Schreier, John D.; Cox, Christopher D.; Fraley, Mark E.; Steen, Justin T.; Lemaire, Wei; Bruno, Joseph G.; Harrell, C. Meacham; Garson, Susan L.; Gotter, Anthony L.; Fox, Steven V.; Stevens, Joanne; Tannenbaum, Pamela L.; Prueksaritanont, Thomayant; Cabalu, ...
Journal:
ChemMedChem
Issue:
Volume 9:Issue 2(2014:Feb.)
Page Start:
241
Record Type:
Journal Article
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3. Discovery of 5′′‐Chloro‐N‐[(5, 6‐dimethoxypyridin‐2‐yl)methyl]‐2, 2′:5′, 3′′‐terpyridine‐3′‐carboxamide (MK‐1064): A Selective Orexin 2 Receptor Antagonist (2‐SORA) for the Treatment of Insomnia. Issue 2 (27th December 2013)

Authors:
Roecker, Anthony J.; Mercer, Swati P.; Schreier, John D.; Cox, Christopher D.; Fraley, Mark E.; Steen, Justin T.; Lemaire, Wei; Bruno, Joseph G.; Harrell, C. Meacham; Garson, Susan L.; Gotter, Anthony L.; Fox, Steven V.; Stevens, Joanne; Tannenbaum, Pamela L.; Prueksaritanont, Thomayant; Cabalu, ...
Journal:
ChemMedChem
Issue:
Volume 9:Issue 2(2014:Feb.)
Page Start:
311
Record Type:
Journal Article
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4. Discovery of diazepane amide DORAs and 2-SORAs enabled by exploration of isosteric quinazoline replacements. Issue 21 (1st November 2015)

Authors:
Roecker, Anthony J.; Mercer, Swati P.; Bergman, Jeffrey M.; Gilbert, Kevin F.; Kuduk, Scott D.; Harrell, C. Meacham; Garson, Susan L.; Fox, Steven V.; Gotter, Anthony L.; Tannenbaum, Pamela L.; Prueksaritanont, Thomayant; Cabalu, Tamara D.; Cui, Donghui; Lemaire, Wei; Winrow, Christopher J.; Reng...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 25:Issue 21(2015)
Page Start:
4992
Record Type:
Journal Article
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5. Discovery of diazepane amide DORAs and 2-SORAs enabled by exploration of isosteric quinazoline replacements. Issue 21 (1st November 2015)

Authors:
Roecker, Anthony J.; Mercer, Swati P.; Bergman, Jeffrey M.; Gilbert, Kevin F.; Kuduk, Scott D.; Harrell, C. Meacham; Garson, Susan L.; Fox, Steven V.; Gotter, Anthony L.; Tannenbaum, Pamela L.; Prueksaritanont, Thomayant; Cabalu, Tamara D.; Cui, Donghui; Lemaire, Wei; Winrow, Christopher J.; Reng...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 25:Issue 21(2015)
Page Start:
4992
Record Type:
Journal Article
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6. Discovery of highly potent and selective orexin 1 receptor antagonists (1-SORAs) suitable for in vivo interrogation of orexin 1 receptor pharmacology. Issue 23 (1st December 2016)

Authors:
Stump, Craig A.; Cooke, Andrew J.; Bruno, Joseph; Cabalu, Tamara D.; Gotter, Anthony L.; Harell, C. Meacham; Kuduk, Scott D.; McDonald, Terrence P.; O'Brien, Julie; Renger, John J.; Williams, Peter D.; Winrow, Christopher J.; Coleman, Paul J.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 23(2016)
Page Start:
5809
Record Type:
Journal Article
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7. Discovery of novel N-1 substituted pyrazolopyrimidinones as potent, selective PDE2 inhibitors. (15th July 2021)

Authors:
Morriello, Gregori J.; Dwyer, Michael P.; Chen, Yili; Ginetti, Anthony T.; Xu, Shimin; Lu, Jun; Abeywickrema, Pravien; Wang, Deping; Crespo, Alejandro; Cabalu, Tamara D.; Wilson, Jonathan E.; Stachel, Shawn J.; Paone, Daniel V.; Sinz, Christopher
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 44(2021)
Page Start:
Record Type:
Journal Article
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8. Discovery of piperidine ethers as selective orexin receptor antagonists (SORAs) inspired by filorexant. Issue 3 (1st February 2015)

Authors:
Raheem, Izzat T.; Breslin, Michael J.; Bruno, Joseph; Cabalu, Tamara D.; Cooke, Andrew; Cox, Christopher D.; Cui, Donghui; Garson, Susan; Gotter, Anthony L.; Fox, Steven V.; Harrell, C. Meacham; Kuduk, Scott D.; Lemaire, Wei; Prueksaritanont, Thomayant; Renger, John J.; Stump, Craig; Tannenbaum, ...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 25:Issue 3(2015)
Page Start:
444
Record Type:
Journal Article
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9. Identification of MK-8133: An orexin-2 selective receptor antagonist with favorable development properties. Issue 12 (15th June 2015)

Authors:
Kuduk, Scott D.; Skudlarek, Jason W.; DiMarco, Christina N.; Bruno, Joseph G.; Pausch, Mark H.; O'Brien, Julie A.; Cabalu, Tamara D.; Stevens, Joanne; Brunner, Joseph; Tannenbaum, Pamela L.; Garson, Susan L.; Savitz, Alan T.; Harrell, Charles M.; Gotter, Anthony L.; Winrow, Christopher J.; Renger...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 25:Issue 12(2015)
Page Start:
2488
Record Type:
Journal Article
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10. Investigation of orexin-2 selective receptor antagonists: Structural modifications resulting in dual orexin receptor antagonists. Issue 6 (15th March 2017)

Authors:
Skudlarek, Jason W.; DiMarco, Christina N.; Babaoglu, Kerim; Roecker, Anthony J.; Bruno, Joseph G.; Pausch, Mark A.; O'Brien, Julie A.; Cabalu, Tamara D.; Stevens, Joanne; Brunner, Joseph; Tannenbaum, Pamela L.; Wuelfing, W. Peter; Garson, Susan L.; Fox, Steven V.; Savitz, Alan T.; Harrell, Charl...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 6(2017)
Page Start:
1364
Record Type:
Journal Article
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