Discovery of diazepane amide DORAs and 2-SORAs enabled by exploration of isosteric quinazoline replacements. Issue 21 (1st November 2015)

• Record Type: Journal Article
• Authors: Roecker, Anthony J.; Mercer, Swati P.; Bergman, Jeffrey M.; Gilbert, Kevin F.; Kuduk, Scott D.; Harrell, C. Meacham; Garson, Susan L.; Fox, Steven V.; Gotter, Anthony L.; Tannenbaum, Pamela L.; Prueksaritanont, Thomayant; Cabalu, Tamara D.; Cui, Donghui; Lemaire, Wei; Winrow, Christopher J.; Renger, John J.; Coleman, Paul J.
• Is Part Of: Bioorganic & medicinal chemistry letters. Volume 25:Issue 21(2015)
• Page Start: 4992
• Page End: 4999
• Publication Date: 2015-11-01
• Subjects: Bioorganic chemistry -- Periodicals; Pharmaceutical chemistry -- Periodicals; 572
• DOI: 10.1016/j.bmcl.2014.12.081
• Languages: English
• ISSNs: 0960-894X

Abstract

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