1. Covalent Inhibitors Allosterically Block the Activation of Rho Family Proteins and Suppress Cancer Cell Invasion. Issue 14 (13th May 2020) Authors: Sun, Zhongya; Zhang, Hao; Zhang, Yuanyuan; Liao, Liping; Zhou, Wen; Zhang, Fengcai; Lian, Fulin; Huang, Jing; Xu, Pan; Zhang, Rukang; Lu, Wenchao; Zhu, Mingrui; Tao, Hongru; Yang, Feng; Ding, Hong; Chen, Shijie; Yue, Liyan; Zhou, Bing; Zhang, Naixia; Tan, Minjia Journal: Advanced science Issue: Volume 7:Issue 14(2020) Page Start: n/a Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Discovery and biological evaluation of thiobarbituric derivatives as potent p300/CBP inhibitors. Issue 20 (1st November 2018) Authors: Lu, Wenchao; Xiong, Huan; Chen, Yu; Wang, Chen; Zhang, Hao; Xu, Pan; Han, Jie; Xiao, Senhao; Ding, Hong; Chen, Zhifeng; Lu, Tian; Wang, Jun; Zhang, Yuanyuan; Yue, Liyan; Liu, Yu-Chih; Zhang, Chenhua; Yang, Yaxi; Jiang, Hualiang; Chen, Kaixian; Zhou, Bing Journal: Bioorganic & medicinal chemistry Issue: Volume 26:Issue 20(2018) Page Start: 5397 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Discovery of novel BET inhibitors by drug repurposing of nitroxoline and its analogues. Issue 44 (31st October 2017) Authors: Jiang, Hao; Xing, Jing; Wang, Chen; Zhang, Hao; Yue, Liyan; Wan, Xiaozhe; Chen, Wei; Ding, Hong; Xie, Yiqian; Tao, Hongru; Chen, Zhifeng; Jiang, Hualiang; Chen, Kaixian; Chen, Shijie; Zheng, Mingyue; Zhang, Yuanyuan; Luo, Cheng Journal: Organic & biomolecular chemistry Issue: Volume 15:Issue 44(2017) Page Start: 9352 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Discovery of novel trimethoxy-ring BRD4 bromodomain inhibitors: AlphaScreen assay, crystallography and cell-based assay12. Issue 6 (22nd May 2017) Authors: Chen, Zhifeng; Zhang, Hao; Liu, Shien; Xie, Yiqian; Jiang, Hao; Lu, Wenchao; Xu, Heng; Yue, Liyan; Zhang, Yuanyuan; Ding, Hong; Zheng, Mingyue; Yu, Kunqian; Chen, Kaixian; Jiang, Hualiang; Luo, Cheng Journal: MedChemComm Issue: Volume 8:Issue 6(2017) Page Start: 1322 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Discovery of trisubstituted nicotinonitrile derivatives as novel human GCN5 inhibitors through AlphaScreen-based high throughput screening. Issue 9 (8th February 2019) Authors: Tao, Hongru; Wang, Jun; Lu, Wenchao; Zhang, Rukang; Xie, Yiqian; Liu, Yu-Chih; Liu, Rongfeng; Yue, Liyan; Chen, Kaixian; Jiang, Hualiang; Zhang, Yuanyuan; Xu, Xiaohui; Luo, Cheng Journal: RSC advances Issue: Volume 9:Issue 9(2019) Page Start: 4917 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Functional interplay between the RK motif and linker segment dictates Oct4–DNA recognition. Issue 9 (13th April 2015) Authors: Kong, Xiangqian; Liu, Jian; Li, Lianchun; Yue, Liyan; Zhang, Lihong; Jiang, Hualiang; Xie, Xin; Luo, Cheng Journal: Nucleic acids research Issue: Volume 43:Issue 9(2015) Page Start: 4381 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. High mobility group box 1 inhibition by BoxA attenuates ovalbumin-induced allergic rhinitis in mice. (17th February 2022) Authors: Yue, Liyan; Dong, Jinhui; Wang, Jianxing; Yin, Xiaoyan; Ren, Xiumin; Xu, Ou; Shan, Chunguang Journal: Autoimmunity Issue: Volume 55:Number 2(2022) Page Start: 118 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Identification of novel small-molecule inhibitors targeting menin–MLL interaction, repurposing the antidiarrheal loperamide. Issue 36 (19th August 2016) Authors: Yue, Liyan; Du, Juanjuan; Ye, Fei; Chen, Zhifeng; Li, Lianchun; Lian, Fulin; Zhang, Bidong; Zhang, Yuanyuan; Jiang, Hualiang; Chen, Kaixian; Li, Yuanchao; Zhou, Bing; Zhang, Naixia; Yang, Yaxi; Luo, Cheng Journal: Organic & biomolecular chemistry Issue: Volume 14:Issue 36(2016) Page Start: 8503 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Inhibition of Autophagy by a Small Molecule through Covalent Modification of the LC3 Protein. (5th November 2021) Authors: Fan, Shijie; Yue, Liyan; Wan, Wei; Zhang, Yuanyuan; Zhang, Bidong; Otomo, Chinatsu; Li, Quanfu; Lin, Tingting; Hu, Junchi; Xu, Pan; Zhu, Mingrui; Tao, Hongru; Chen, Zhifeng; Li, Lianchun; Ding, Hong; Yao, Zhiyi; Lu, Junyan; Wen, Yi; Zhang, Naixia; Tan, Minjia Journal: Angewandte Chemie Issue: Volume 133:Number 50(2021) Page Start: 26309 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. Inhibition of Autophagy by a Small Molecule through Covalent Modification of the LC3 Protein. Issue 50 (5th November 2021) Authors: Fan, Shijie; Yue, Liyan; Wan, Wei; Zhang, Yuanyuan; Zhang, Bidong; Otomo, Chinatsu; Li, Quanfu; Lin, Tingting; Hu, Junchi; Xu, Pan; Zhu, Mingrui; Tao, Hongru; Chen, Zhifeng; Li, Lianchun; Ding, Hong; Yao, Zhiyi; Lu, Junyan; Wen, Yi; Zhang, Naixia; Tan, Minjia Journal: Angewandte Chemie international edition Issue: Volume 60:Issue 50(2021) Page Start: 26105 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗