1. 'Turn On/Off' fluorescence probe for the screening of unactivated Bruton's tyrosine kinase. Issue 10 (15th May 2015) Authors: Kawahata, Wataru; Asami, Tokiko; Fujii, Ikuo; Sawa, Masaaki Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 10(2015) Page Start: 2141 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. 'Turn On/Off' fluorescence probe for the screening of unactivated Bruton's tyrosine kinase. Issue 10 (15th May 2015) Authors: Kawahata, Wataru; Asami, Tokiko; Fujii, Ikuo; Sawa, Masaaki Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 10(2015) Page Start: 2141 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. 5Z-7-Oxozeaenol covalently binds to MAP2K7 at Cys218 in an unprecedented manner. Issue 3 (1st February 2015) Authors: Sogabe, Yuri; Matsumoto, Takashi; Hashimoto, Takuma; Kirii, Yasuyuki; Sawa, Masaaki; Kinoshita, Takayoshi Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 3(2015) Page Start: 593 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. A promiscuous kinase inhibitor delineates the conspicuous structural features of protein kinase CK2a1. Issue 7 (8th July 2019) Authors: Tsuyuguchi, Masato; Nakaniwa, Tetsuko; Sawa, Masaaki; Nakanishi, Isao; Kinoshita, Takayoshi Journal: Acta crystallographica Issue: Volume 75:Issue 7(2019:Jul.) Page Start: 515 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. An isoform-selective inhibitor of tropomyosin receptor kinase A behaves as molecular glue. Issue 1 (1st January 2020) Authors: Furuya, Noritaka; Momose, Takaki; Katsuno, Kenji; Fushimi, Nobuhiko; Muranaka, Hideyuki; Handa, Chiaki; Sawa, Masaaki; Ozawa, Tomonaga; Kinoshita, Takayoshi Journal: Bioorganic & medicinal chemistry letters Issue: Volume 30:Issue 1(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Compound Selectivity and Target Residence Time of Kinase Inhibitors Studied with Surface Plasmon Resonance. Issue 4 (17th February 2017) Authors: Willemsen-Seegers, Nicole; Uitdehaag, Joost C.M.; Prinsen, Martine B.W.; de Vetter, Judith R.F.; de Man, Jos; Sawa, Masaaki; Kawase, Yusuke; Buijsman, Rogier C.; Zaman, Guido J.R. Journal: Journal of molecular biology Issue: Volume 429:Issue 4(2017) Page Start: 574 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Design and synthesis of novel pyrimidine analogs as highly selective, non-covalent BTK inhibitors. Issue 2 (15th January 2018) Authors: Kawahata, Wataru; Asami, Tokiko; Irie, Takayuki; Sawa, Masaaki Journal: Bioorganic & medicinal chemistry letters Issue: Volume 28:Issue 2(2018) Page Start: 145 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Identification of an allosteric and Smad3-selective inhibitor of p38αMAPK using a substrate-based approach. (1st July 2021) Authors: Nagao, Haruna; Kitagawa, Daisuke; Nakajima, Fumio; Sawa, Masaaki; Kinoshita, Takayoshi Journal: Bioorganic & medicinal chemistry letters Issue: Volume 43(2021) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Structure of mitogen‐activated protein kinase kinase 1 in the DFG‐out conformation. Issue 12 (25th November 2021) Authors: Nakae, Setsu; Kitamura, Maho; Fujiwara, Daisuke; Sawa, Masaaki; Shirai, Tsuyoshi; Fujii, Ikuo; Tada, Toshiji Journal: Acta crystallographica Issue: Volume 77:Issue 12(2021) Page Start: 459 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. Targeting the Wnt signaling pathway in colorectal cancer. (2nd April 2016) Authors: Sawa, Masaaki; Masuda, Mari; Yamada, Tesshi Journal: Expert opinion on therapeutic targets Issue: Volume 20:Number 4(2016:Apr.) Page Start: 419 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗