1. A combined ligand- and structure-based approach for the identification of rilmenidine-derived compounds which synergize the antitumor effects of doxorubicin. Issue 14 (15th July 2016) Authors: Vucicevic, Jelica; Srdic-Rajic, Tatjana; Pieroni, Marco; Laurila, Jonne M.M.; Perovic, Vladimir; Tassini, Sabrina; Azzali, Elisa; Costantino, Gabriele; Glisic, Sanja; Agbaba, Danica; Scheinin, Mika; Nikolic, Katarina; Radi, Marco; Veljkovic, Nevena Journal: Bioorganic & medicinal chemistry Issue: Volume 24:Issue 14(2016) Page Start: 3174 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Adjuvant therapies against tuberculosis: discovery of a 2-aminothiazole targeting Mycobacterium tuberculosis energetics. (September 2018) Authors: Machado, Diana; Azzali, Elisa; Couto, Isabel; Costantino, Gabriele; Pieroni, Marco; Viveiros, Miguel Journal: Future microbiology Issue: Volume 13:Number 12(2018) Page Start: 1383 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Cover Picture: Discovery of New Potential Anti‐Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target‐Focused Repurposing Approaches (ChemMedChem 17/2016). (6th September 2016) Authors: Annunziato, Giannamaria; Angeli, Andrea; D'Alba, Francesca; Bruno, Agostino; Pieroni, Marco; Vullo, Daniela; De Luca, Viviana; Capasso, Clemente; Supuran, Claudiu T.; Costantino, Gabriele Journal: ChemMedChem Issue: Volume 11:Number 17(2016) Page Start: 1876 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Crystal structure of Aspergillus fumigatus AroH, an aromatic amino acid aminotransferase. Issue 2 (16th September 2021) Authors: Spizzichino, Sharon; Pampalone, Gioena; Dindo, Mirco; Bruno, Agostino; Romani, Luigina; Cutruzzolà, Francesca; Zelante, Teresa; Pieroni, Marco; Cellini, Barbara; Giardina, Giorgio Journal: Proteins Issue: Volume 90:Issue 2(2022) Page Start: 435 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Cyclopropane derivatives as potential human serine racemase inhibitors: unveiling novel insights into a difficult target. (3rd July 2016) Authors: Beato, Claudia; Pecchini, Chiara; Cocconcelli, Chiara; Campanini, Barbara; Marchetti, Marialaura; Pieroni, Marco; Mozzarelli, Andrea; Costantino, Gabriele Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 31(2016.)Supplement 4 Page Start: 645 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Cyclopropane-1, 2-dicarboxylic acids as new tools for the biophysical investigation of O-acetylserine sulfhydrylases by fluorimetric methods and saturation transfer difference (STD) NMR. (4th November 2016) Authors: Annunziato, Giannamaria; Pieroni, Marco; Benoni, Roberto; Campanini, Barbara; Pertinhez, Thelma A.; Pecchini, Chiara; Bruno, Agostino; Magalhães, Joana; Bettati, Stefano; Franko, Nina; Mozzarelli, Andrea; Costantino, Gabriele Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 31(2016.)Supplement 4 Page Start: 78 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Cycloserine enantiomers are reversible inhibitors of human alanine:glyoxylate aminotransferase: implications for Primary Hyperoxaluria type 1. Issue 24 (20th December 2019) Authors: Dindo, Mirco; Grottelli, Silvia; Annunziato, Giannamaria; Giardina, Giorgio; Pieroni, Marco; Pampalone, Gioena; Faccini, Andrea; Cutruzzolà, Francesca; Laurino, Paola; Costantino, Gabriele; Cellini, Barbara Journal: Biochemical journal Issue: Volume 476:Issue 24(2019) Page Start: 3751 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Discovering a new class of antifungal agents that selectively inhibits microbial carbonic anhydrases. (1st January 2018) Authors: Annunziato, Giannamaria; Giovati, Laura; Angeli, Andrea; Pavone, Marialaura; Del Prete, Sonia; Pieroni, Marco; Capasso, Clemente; Bruno, Agostino; Conti, Stefania; Magliani, Walter; Supuran, Claudiu T.; Costantino, Gabriele Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 33:Number 1(2018) Page Start: 1537 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Discovery of New Potential Anti‐Infective Compounds Based on Carbonic Anhydrase Inhibitors by Rational Target‐Focused Repurposing Approaches. (15th June 2016) Authors: Annunziato, Giannamaria; Angeli, Andrea; D'Alba, Francesca; Bruno, Agostino; Pieroni, Marco; Vullo, Daniela; De Luca, Viviana; Capasso, Clemente; Supuran, Claudiu T.; Costantino, Gabriele Journal: ChemMedChem Issue: Volume 11:Number 17(2016) Page Start: 1904 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. Discovery of novel fragments inhibiting O-acetylserine sulphhydrylase by combining scaffold hopping and ligand–based drug design. (1st January 2018) Authors: Magalhães, Joana; Franko, Nina; Annunziato, Giannamaria; Welch, Martin; Dolan, Stephen K.; Bruno, Agostino; Mozzarelli, Andrea; Armao, Stefano; Jirgensons, Aigars; Pieroni, Marco; Costantino, Gabriele; Campanini, Barbara Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 33:Number 1(2018) Page Start: 1444 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗