1. C-3 benzoic acid derivatives of C-3 deoxybetulinic acid and deoxybetulin as HIV-1 maturation inhibitors. Issue 8 (15th April 2016) Authors: Liu, Zheng; Swidorski, Jacob J.; Nowicka-Sans, Beata; Terry, Brian; Protack, Tricia; Lin, Zeyu; Samanta, Himadri; Zhang, Sharon; Li, Zhufang; Parker, Dawn D.; Rahematpura, Sandhya; Jenkins, Susan; Beno, Brett R.; Krystal, Mark; Meanwell, Nicholas A.; Dicker, Ira B.; Regueiro-Ren, Alicia Journal: Bioorganic & medicinal chemistry Issue: Volume 24:Issue 8(2016) Page Start: 1757 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Design and exploration of C-3 benzoic acid bioisosteres and alkyl replacements in the context of GSK3532795 (BMS-955176) that exhibit broad spectrum HIV-1 maturation inhibition. (15th March 2021) Authors: Swidorski, Jacob J.; Jenkins, Susan; Hanumegowda, Umesh; Parker, Dawn D.; Beno, Brett R.; Protack, Tricia; Ng, Alicia; Gupta, Anuradha; Shanmugam, Yoganand; Dicker, Ira B.; Krystal, Mark; Meanwell, Nicholas A.; Regueiro-Ren, Alicia Journal: Bioorganic & medicinal chemistry letters Issue: Volume 36(2021) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Design, synthesis and SAR study of novel C2-pyrazolopyrimidine amides and amide isosteres as allosteric integrase inhibitors. Issue 21 (1st November 2020) Authors: Patel, Manoj; Cianci, Christopher; Allard, Christopher W.; Parker, Dawn D.; Simmermacher, Jean; Jenkins, Susan; Mcauliffe, Brian; Minassian, Beatrice; Discotto, Linda; Krystal, Mark; Meanwell, Nicholas A.; Naidu, B. Narasimhulu Journal: Bioorganic & medicinal chemistry letters Issue: Volume 30:Issue 21(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Discovery and preclinical evaluation of potent, orally bioavailable, metabolically stable cyclopropylindolobenzazepine acylsulfonamides as thumb site 1 inhibitors of the hepatitis c virus NS5B RNA-dependent, RNA polymerase. Issue 3 (1st February 2016) Authors: Hewawasam, Piyasena; Tu, Yong; Gao, Min; Hanumegowda, Umesh; Knipe, Jay; Lemm, Julie A.; Parker, Dawn D.; Rigat, Karen L.; Roberts, Susan B.; Meanwell, Nicholas A.; Kadow, John F. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 3(2016) Page Start: 936 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Discovery and preclinical evaluation of potent, orally bioavailable, metabolically stable cyclopropylindolobenzazepine acylsulfonamides as thumb site 1 inhibitors of the hepatitis c virus NS5B RNA-dependent, RNA polymerase. Issue 3 (1st February 2016) Authors: Hewawasam, Piyasena; Tu, Yong; Gao, Min; Hanumegowda, Umesh; Knipe, Jay; Lemm, Julie A.; Parker, Dawn D.; Rigat, Karen L.; Roberts, Susan B.; Meanwell, Nicholas A.; Kadow, John F. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 3(2016) Page Start: 936 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Inhibitors of HIV-1 attachment: The discovery and structure–activity relationships of tetrahydroisoquinolines as replacements for the piperazine benzamide in the 3-glyoxylyl 6-azaindole pharmacophore. Issue 1 (1st January 2016) Authors: Swidorski, Jacob J.; Liu, Zheng; Yin, Zhiwei; Wang, Tao; Carini, David J.; Rahematpura, Sandhya; Zheng, Ming; Johnson, Kim; Zhang, Sharon; Lin, Pin-Fang; Parker, Dawn D.; Li, Wenying; Meanwell, Nicholas A.; Hamann, Lawrence G.; Regueiro-Ren, Alicia Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 1(2016) Page Start: 160 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Inhibitors of HIV-1 maturation: Development of structure–activity relationship for C-28 amides based on C-3 benzoic acid-modified triterpenoids. Issue 8 (15th April 2016) Authors: Swidorski, Jacob J.; Liu, Zheng; Sit, Sing-Yuen; Chen, Jie; Chen, Yan; Sin, Ny; Venables, Brian L.; Parker, Dawn D.; Nowicka-Sans, Beata; Terry, Brian J.; Protack, Tricia; Rahematpura, Sandhya; Hanumegowda, Umesh; Jenkins, Susan; Krystal, Mark; Dicker, Ira B.; Meanwell, Nicholas A.; Regueiro-Ren,... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 8(2016) Page Start: 1925 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Scaffold modifications to the 4-(4, 4-dimethylpiperidinyl) 2, 6-dimethylpyridinyl class of HIV-1 allosteric integrase inhibitors. (1st August 2022) Authors: Parcella, Kyle; Patel, Manoj; Tu, Yong; Eastman, Kyle; Peese, Kevin; Gillis, Eric; Belema, Makonen; Dicker, Ira B.; McAuliffe, Brian; Ding, Bo; Falk, Paul; Simmermacher, Jean; Parker, Dawn D.; Sivaprakasam, Prasanna; Khan, Javed A.; Kish, Kevin; Lewis, Hal; Hanumegowda, Umesh; Jenkins, Susan; Kad... Journal: Bioorganic & medicinal chemistry Issue: Volume 67(2022) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Synthesis and evaluation of C2-carbon-linked heterocyclic-5-hydroxy-6-oxo-dihydropyrimidine-4-carboxamides as HIV-1 integrase inhibitors. Issue 3 (1st February 2015) Authors: Naidu, B. Narasimhulu; Sorenson, Margaret E.; Patel, Manoj; Ueda, Yasutsugu; Banville, Jacques; Beaulieu, Francis; Bollini, Sagarika; Dicker, Ira B.; Higley, Helen; Lin, Zeyu; Pajor, Lori; Parker, Dawn D.; Terry, Brian J.; Zheng, Ming; Martel, Alain; Meanwell, Nicholas A.; Krystal, Mark; Walker, ... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 3(2015) Page Start: 717 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. The design, synthesis and structure-activity relationships associated with C28 amine-based betulinic acid derivatives as inhibitors of HIV-1 maturation. Issue 9 (15th May 2018) Authors: Chen, Yan; Sit, Sing-Yuen; Chen, Jie; Swidorski, Jacob J.; Liu, Zheng; Sin, Ny; Venables, Brian L.; Parker, Dawn D.; Nowicka-Sans, Beata; Lin, Zeyu; Li, Zhufang; Terry, Brian J.; Protack, Tricia; Rahematpura, Sandhya; Hanumegowda, Umesh; Jenkins, Susan; Krystal, Mark; Dicker, Ira D.; Meanwell, Ni... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 28:Issue 9(2018) Page Start: 1550 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗