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Author/Creator Olson, Richard E.

1. An amide-based sulfenamide prodrug of gamma secretase inhibitor BMS–708163 delivers parent drug from an oral conventional solid dosage form in male beagle dog. Issue 3 (1st February 2020)

Authors:
Guarino, Victor R.; Olson, Richard E.; Everlof, J. Gerry; Wang, Nenghui; McDonald, Ivar; Haskell, Roy; Clarke, Wendy; Lentz, Kimberley A.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 30:Issue 3(2020)
Page Start:
Record Type:
Journal Article
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3. Design and synthesis of a novel series of (1′S, 2R, 4′S)-3H-4′-azaspiro[benzo[4, 5]imidazo[2, 1-b]oxazole-2, 2′-bicyclo[2.2.2]octanes] with high affinity for the α7 neuronal nicotinic receptor. Issue 22 (15th November 2017)

Authors:
Cook, James; Zusi, F. Christopher; Hill, Matthew D.; Fang, Haiquan; Pearce, Bradley; Park, Hyunsoo; Gallagher, Lizbeth; McDonald, Ivar M.; Bristow, Linda; Macor, John E.; Olson, Richard E.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 22(2017)
Page Start:
5002
Record Type:
Journal Article
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4. Design and synthesis of a novel series of 4-heteroarylamino-1′-azaspiro[oxazole-5, 3′-bicyclo[2.2.2]octanes as α7 nicotinic receptor agonists 2. Development of 4-heteroaryl SAR. Issue 5 (1st March 2017)

Authors:
Iwuagwu, Christiana; King, Dalton; McDonald, Ivar M.; Cook, James; Zusi, F. Christopher; Hill, Matthew D.; Mate, Robert A.; Fang, Haiquan; Knox, Ronald; Gallagher, Lizbeth; Post-Munson Amy Easton, Debra; Miller, Regina; Benitex, Yulia; Siuciak, Judy; Lodge, Nicholas; Zaczek, Robert; Morgan, Danie...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 5(2017)
Page Start:
1261
Record Type:
Journal Article
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5. Development of spiroguanidine-derived α7 neuronal nicotinic receptor partial agonists. Issue 3 (1st February 2017)

Authors:
Hill, Matthew D.; Fang, Haiquan; Digavalli, Sivarao V.; Healy, Francine L.; Gallagher, Lizbeth; Post-Munson, Debra; Chen, Ping; Natale, Joanne; Benitex, Yulia; Morgan, Daniel; Lodge, Nicholas; Bristow, Linda; Macor, John E.; Olson, Richard E.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 3(2017)
Page Start:
578
Record Type:
Journal Article
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6. Identification and Preclinical Pharmacology of the γ-Secretase Modulator BMS-869780. (7th July 2014)

Authors:
Toyn, Jeremy H.; Thompson, Lorin A.; Lentz, Kimberley A.; Meredith, Jere E.; Burton, Catherine R.; Sankaranararyanan, Sethu; Guss, Valerie; Hall, Tracey; Iben, Lawrence G.; Krause, Carol M.; Krause, Rudy; Lin, Xu-Alan; Pierdomenico, Maria; Polson, Craig; Robertson, Alan S.; Denton, R. Rex; Grace,...
Other Names:
Perry George Academic Editor.
Journal:
International journal of alzheimer's disease
Issue:
Volume 2014(2014)
Page Start:
Record Type:
Journal Article
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7. Macrocyclic prolinyl acyl guanidines as inhibitors of β-secretase (BACE). Issue 22 (15th November 2015)

Authors:
Boy, Kenneth M.; Guernon, Jason M.; Wu, Yong-Jin; Zhang, Yunhui; Shi, Joe; Zhai, Weixu; Zhu, Shirong; Gerritz, Samuel W.; Toyn, Jeremy H.; Meredith, Jere E.; Barten, Donna M.; Burton, Catherine R.; Albright, Charles F.; Good, Andrew C.; Grace, James E.; Lentz, Kimberley A.; Olson, Richard E.; Mac...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 25:Issue 22(2015)
Page Start:
5040
Record Type:
Journal Article
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10. Synthesis of carbon‐14 and stable isotope labeled Avagacestat: a novel gamma secretase inhibitor for the treatment of Alzheimer's disease. (5th September 2014)

Authors:
Burrell, Richard C.; Easter, John A.; Cassidy, Michael P.; Gillman, Kevin W.; Olson, Richard E.; Bonacorsi, Samuel J.
Journal:
Journal of labelled compounds & radiopharmaceuticals
Issue:
Volume 57:Number 10(2014)
Page Start:
600
Record Type:
Journal Article
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