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Author/Creator Niswender, Colleen M.

2. Acyl dihydropyrazolo[1, 5-a]pyrimidinones as metabotropic glutamate receptor 5 positive allosteric modulators. Issue 22 (15th November 2015)

Authors:
Malosh, Chrysa; Turlington, Mark; Bridges, Thomas M.; Rook, Jerri M.; Noetzel, Meredith J.; Vinson, Paige N.; Steckler, Thomas; Lavreysen, Hilde; Mackie, Claire; Bartolomé-Nebreda, José M.; Conde-Ceide, Susana; Martínez-Viturro, Carlos M.; Piedrafita, María; Sánchez-Casado, M. Rosa; Macdonald, Gr...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 25:Issue 22(2015)
Page Start:
5115
Record Type:
Journal Article
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3. Application of Parallel Multiparametric Cell-Based FLIPR Detection Assays for the Identification of Modulators of the Muscarinic Acetylcholine Receptor 4 (M4). (August 2015)

Authors:
Smith, Emery; Chase, Peter; Niswender, Colleen M.; Utley, Thomas J.; Sheffler, Douglas J.; Noetzel, Meredith J.; Lamsal, Atin; Wood, Michael R.; Conn, P. Jeffrey; Lindsley, Craig W.; Madoux, Franck; Acosta, Mary; Scampavia, Louis; Spicer, Timothy; Hodder, Peter
Journal:
Journal of biomolecular screening
Issue:
Volume 20:Number 7(2015)
Page Start:
858
Record Type:
Journal Article
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4. Challenges in the development of an M4 PAM in vivo tool compound: The discovery of VU0467154 and unexpected DMPK profiles of close analogs. Issue 2 (15th January 2017)

Authors:
Wood, Michael R.; Noetzel, Meredith J.; Poslusney, Michael S.; Melancon, Bruce J.; Tarr, James C.; Lamsal, Atin; Chang, Sichen; Luscombe, Vincent B.; Weiner, Rebecca L.; Cho, Hyekyung P.; Bubser, Michael; Jones, Carrie K.; Niswender, Colleen M.; Wood, Michael W.; Engers, Darren W.; Brandon, Nicho...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 2(2017)
Page Start:
171
Record Type:
Journal Article
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5. Challenges in the development of an M4 PAM preclinical candidate: The discovery, SAR, and biological characterization of a series of azetidine-derived tertiary amides. Issue 23 (1st December 2017)

Authors:
Tarr, James C.; Wood, Michael R.; Noetzel, Meredith J.; Melancon, Bruce J.; Lamsal, Atin; Luscombe, Vincent B.; Rodriguez, Alice L.; Byers, Frank W.; Chang, Sichen; Cho, Hyekyung P.; Engers, Darren W.; Jones, Carrie K.; Niswender, Colleen M.; Wood, Michael W.; Brandon, Nicholas J.; Duggan, Mark E...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 23(2017)
Page Start:
5179
Record Type:
Journal Article
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6. Challenges in the development of an M4 PAM preclinical candidate: The discovery, SAR, and in vivo characterization of a series of 3-aminoazetidine-derived amides. Issue 13 (1st July 2017)

Authors:
Tarr, James C.; Wood, Michael R.; Noetzel, Meredith J.; Bertron, Jeanette L.; Weiner, Rebecca L.; Rodriguez, Alice L.; Lamsal, Atin; Byers, Frank W.; Chang, Sichen; Cho, Hyekyung P.; Jones, Carrie K.; Niswender, Colleen M.; Wood, Michael W.; Brandon, Nicholas J.; Duggan, Mark E.; Conn, P. Jeffrey...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 13(2017)
Page Start:
2990
Record Type:
Journal Article
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7. Cognitive enhancement and antipsychotic-like activity following repeated dosing with the selective M4 PAM VU0467154. (January 2018)

Authors:
Gould, Robert W.; Grannan, Michael D.; Gunter, Barak W.; Ball, Jacob; Bubser, Michael; Bridges, Thomas M.; Wess, Jurgen; Wood, Michael W.; Brandon, Nicholas J.; Duggan, Mark E.; Niswender, Colleen M.; Lindsley, Craig W.; Conn, P. Jeffrey; Jones, Carrie K.
Journal:
Neuropharmacology
Issue:
Volume 128(2018)
Page Start:
492
Record Type:
Journal Article
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8. Corrigendum to "Challenges in the development of an M4 PAM preclinical candidate: The discovery, SAR, and biological characterization of a series of azetidine-derived tertiary amides" [Bioorg. Med. Chem. Lett. 27(23) (2017) 5179–5184]. Issue 17 (15th September 2018)

Authors:
Tarr, James C.; Wood, Michael R.; Noetzel, Meredith J.; Melancon, Bruce J.; Lamsal, Atin; Luscombe, Vincent B.; Rodriguez, Alice L.; Byers, Frank W.; Chang, Sichen; Cho, Hyekyung P.; Engers, Darren W.; Jones, Carrie K.; Niswender, Colleen M.; Wood, Michael W.; Brandon, Nicholas J.; Duggan, Mark E...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 28:Issue 17(2018)
Page Start:
3014
Record Type:
Journal Article
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9. Corrigendum to "Novel GlyT1 inhibitor chemotypes by scaffold hopping. Part 2: Development of a [3.3.0]-based series and other piperidine bioisosteres" [Bioorg. Med. Chem. Lett. 24 (2014) 1062–1066]. Issue 9 (1st May 2017)

Authors:
Sheffler, Douglas J.; Nedelcovych, Michael T.; Williams, Richard; Turner, Stephen C.; Duerk, Brittany B.; Robbins, Megan R.; Jadhav, Sataya B.; Niswender, Colleen M.; Jones, Carrie K.; Conn, P. Jeffrey; Nathan Daniels, R.; Lindsley, Craig W.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 9(2017)
Page Start:
2079
Record Type:
Journal Article
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10. Development and profiling of mGlu7 NAMs with a range of saturable inhibition of agonist responses in vitro. (15th October 2022)

Authors:
Reed, Carson W.; Rodriguez, Alice L.; Kalbfleisch, Jacob J.; Seto, Mabel; Jenkins, Matthew T.; Blobaum, Anna L.; Chang, Sichen; Lindsley, Craig W.; Niswender, Colleen M.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 74(2022)
Page Start:
Record Type:
Journal Article
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