1. A metal-catalyzed enyne-cyclization step for the synthesis of bi- and tricyclic scaffolds amenable to molecular library production. Issue 29 (30th June 2016) Authors: Wu, Peng; Petersen, Michael Åxman; Cohrt, A. Emil; Petersen, Rico; Morgentin, Rémy; Lemoine, Hugues; Roche, Carine; Willaume, Anthony; Clausen, Mads H.; Nielsen, Thomas E. Journal: Organic & biomolecular chemistry Issue: Volume 14:Issue 29(2016) Page Start: 6947 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Discovery of 1-(4-(5-(5-amino-6-(5-tert-butyl-1, 3, 4-oxadiazol-2-yl)pyrazin-2-yl)-1-ethyl-1, 2, 4-triazol-3-yl)piperidin-1-yl)-3-hydroxypropan-1-one (AZD8835): A potent and selective inhibitor of PI3Kα and PI3Kδ for the treatment of cancers. Issue 22 (15th November 2015) Authors: Barlaam, Bernard; Cosulich, Sabina; Delouvrié, Bénédicte; Ellston, Rebecca; Fitzek, Martina; Germain, Hervé; Green, Stephen; Hancox, Urs; Harris, Craig S.; Hudson, Kevin; Lambert-van der Brempt, Christine; Lebraud, Honorine; Magnien, Françoise; Lamorlette, Maryannick; Le Griffon, Antoine; Morgent... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 22(2015) Page Start: 5155 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Discovery of a series of 8-(1-phenylpyrrolidin-2-yl)-6-carboxamide-2-morpholino-4H-chromen-4-one as PI3Kβ/δ inhibitors for the treatment of PTEN-deficient tumours. Issue 9 (1st May 2017) Authors: Barlaam, Bernard; Cosulich, Sabina; Degorce, Sébastien; Ellston, Rebecca; Fitzek, Martina; Green, Stephen; Hancox, Urs; Lambert-van der Brempt, Christine; Lohmann, Jean-Jacques; Maudet, Mickaël; Morgentin, Rémy; Plé, Patrick; Ward, Lara; Warin, Nicolas Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 9(2017) Page Start: 1949 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Discovery of a series of 8-(2, 3-dihydro-1, 4-benzoxazin-4-ylmethyl)-2-morpholino-4-oxo-chromene-6-carboxamides as PI3Kβ/δ inhibitors for the treatment of PTEN-deficient tumours. Issue 9 (1st May 2016) Authors: Barlaam, Bernard; Cosulich, Sabina; Degorce, Sébastien; Fitzek, Martina; Green, Stephen; Hancox, Urs; Lambert-van der Brempt, Christine; Lohmann, Jean-Jacques; Maudet, Mickaël; Morgentin, Rémy; Péru, Aurélien; Plé, Patrick; Saleh, Twana; Ward, Lara; Warin, Nicolas Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 9(2016) Page Start: 2318 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Petasis/Diels–Alder/Cyclization Cascade Reactions for the Generation of Scaffolds with Multiple Stereogenic Centers and Orthogonal Handles for Library Production. Issue 36 (15th June 2018) Authors: Flagstad, Thomas; Azevedo, Carlos M. G.; Min, Geanna; Willaume, Anthony; Morgentin, Rémy; Nielsen, Thomas E.; Clausen, Mads H. Journal: European journal of organic chemistry Issue: Issue 36(2018) Page Start: 5023 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Petasis/Diels–Alder/Cyclization Cascade Reactions for the Generation of Scaffolds with Multiple Stereogenic Centers and Orthogonal Handles for Library Production. Issue 46 (13th December 2018) Authors: Flagstad, Thomas; Azevedo, Carlos M. G.; Min, Geanna; Willaume, Anthony; Morgentin, Rémy; Nielsen, Thomas E.; Clausen, Mads H. Journal: European journal of organic chemistry Issue: Issue 46(2018) Page Start: 6596 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Realisation of small molecule libraries based on frameworks distantly related to natural products. Issue 17 (12th April 2018) Authors: Aimon, Anthony; Karageorgis, George; Masters, Jacob; Dow, Mark; Craven, Philip G. E.; Ohsten, Martin; Willaume, Anthony; Morgentin, Rémy; Ruiz-Llamas, Nicolas; Lemoine, Hugues; Kalliokoski, Tuomo; Eatherton, Andrew J.; Foley, Daniel J.; Marsden, Stephen P.; Nelson, Adam Journal: Organic & biomolecular chemistry Issue: Volume 16:Issue 17(2018) Page Start: 3160 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Squaramides as novel class I and IIB histone deacetylase inhibitors for topical treatment of cutaneous t-cell lymphoma. Issue 17 (15th September 2018) Authors: Fournier, Jean-François; Bhurruth-Alcor, Yushma; Musicki, Branislav; Aubert, Jérome; Aurelly, Michèle; Bouix-Peter, Claire; Bouquet, Karinne; Chantalat, Laurent; Delorme, Marion; Drean, Bénédicte; Duvert, Gwenaelle; Fleury-Bregeot, Nicolas; Gauthier, Blanche; Grisendi, Karine; Harris, Craig S.; H... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 28:Issue 17(2018) Page Start: 2985 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Synthesis of 1, 4, 5 trisubstituted γ-lactams via a 3-component cascade reaction. Issue 11 (1st June 2015) Authors: Petersen, Michael Åxman; Mortensen, Michael A.; Cohrt, A. Emil; Petersen, Rico; Wu, Peng; Fleury-Brégeot, Nicolas; Morgentin, Rémy; Lardy, Claude; Nielsen, Thomas E.; Clausen, Mads H. Journal: Bioorganic & medicinal chemistry Issue: Volume 23:Issue 11(2015) Page Start: 2695 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. Tandem Mannich/Diels–Alder reactions for the synthesis of indole compound libraries. Issue 52 (12th May 2016) Authors: Wu, Peng; Petersen, Michael Åxman; Petersen, Rico; Flagstad, Thomas; Guilleux, Rachel; Ohsten, Martin; Morgentin, Rémy; Nielsen, Thomas E.; Clausen, Mads H. Journal: RSC advances Issue: Volume 6:Issue 52(2016) Page Start: 46654 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗