1. 4-Aryliden-2-methyloxazol-5(4H)-one as a new scaffold for selective reversible MAGL inhibitors. (2nd January 2016) Authors: Granchi, Carlotta; Rizzolio, Flavio; Bordoni, Vittorio; Caligiuri, Isabella; Manera, Clementina; Macchia, Marco; Minutolo, Filippo; Martinelli, Adriano; Giordano, Antonio; Tuccinardi, Tiziano Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 31:Number 1(2016:Feb.) Page Start: 137 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. A patent review of Monoacylglycerol Lipase (MAGL) inhibitors (2013-2017). (2nd December 2017) Authors: Granchi, Carlotta; Caligiuri, Isabella; Minutolo, Filippo; Rizzolio, Flavio; Tuccinardi, Tiziano Journal: Expert opinion on therapeutic patents Issue: Volume 27:Number 12(2017:Dec.) Page Start: 1341 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. A specific inhibitor of lactate dehydrogenase overcame the resistance toward gemcitabine in hypoxic mesothelioma cells, and modulated the expression of the human equilibrative transporter-1. (1st December 2016) Authors: Giovannetti, Elisa; Leon, Leticia G.; Gómez, Valentina E.; Zucali, Paolo A.; Minutolo, Filippo; Peters, Godefridus J. Journal: Nucleosides, nucleotides & nucleic acids Issue: Volume 35:Number 10/12(2016) Page Start: 643 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. A Virtual Screening Study for Lactate Dehydrogenase 5 Inhibitors by Using a Pharmacophore‐based Approach. Issue 8 (15th June 2016) Authors: Tuccinardi, Tiziano; Poli, Giulio; Corchia, Isacco; Granchi, Carlotta; Lapillo, Margherita; Macchia, Marco; Minutolo, Filippo; Ortore, Gabriella; Martinelli, Adriano Journal: Molecular informatics Issue: Volume 35:Issue 8/9(2016) Page Start: 434 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. An Update on Patents Covering Agents That Interfere with the Cancer Glycolytic Cascade. (9th October 2018) Authors: Fortunato, Serena; Bononi, Giulia; Granchi, Carlotta; Minutolo, Filippo Journal: ChemMedChem Issue: Volume 13:Number 21(2018) Page Start: 2251 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. An updated patent review of monoacylglycerol lipase (MAGL) inhibitors (2018-present). (1st February 2021) Authors: Bononi, Giulia; Poli, Giulio; Rizzolio, Flavio; Tuccinardi, Tiziano; Macchia, Marco; Minutolo, Filippo; Granchi, Carlotta Journal: Expert opinion on therapeutic patents Issue: Volume 31:Number 2(2021) Page Start: 153 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Binding investigation and preliminary optimisation of the 3-amino-1, 2, 4-triazin-5(2H)-one core for the development of new Fyn inhibitors. (1st January 2018) Authors: Poli, Giulio; Lapillo, Margherita; Granchi, Carlotta; Caciolla, Jessica; Mouawad, Nayla; Caligiuri, Isabella; Rizzolio, Flavio; Langer, Thierry; Minutolo, Filippo; Tuccinardi, Tiziano Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 33:Number 1(2018) Page Start: 956 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Computationally driven discovery of phenyl(piperazin-1-yl)methanone derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors. (1st January 2019) Authors: Poli, Giulio; Lapillo, Margherita; Jha, Vibhu; Mouawad, Nayla; Caligiuri, Isabella; Macchia, Marco; Minutolo, Filippo; Rizzolio, Flavio; Tuccinardi, Tiziano; Granchi, Carlotta Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 34:Number 1(2019) Page Start: 589 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Cyclic Ketoximes as Estrogen Receptor β Selective Agonists. (2nd May 2016) Authors: Granchi, Carlotta; Lapillo, Margherita; Spena, Concetta Russo; Rizzolio, Flavio; Tuccinardi, Tiziano; Martin, Teresa A.; Carlson, Kathryn E.; Katzenellenbogen, John A.; Minutolo, Filippo Journal: ChemMedChem Issue: Volume 11:Number 16(2016) Page Start: 1752 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. Development of terphenyl-2-methyloxazol-5(4H)-one derivatives as selective reversible MAGL inhibitors. (1st January 2017) Authors: Granchi, Carlotta; Caligiuri, Isabella; Bertelli, Eleonora; Poli, Giulio; Rizzolio, Flavio; Macchia, Marco; Martinelli, Adriano; Minutolo, Filippo; Tuccinardi, Tiziano Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 32:Number 1(2017) Page Start: 1240 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗