1. 4-Aryliden-2-methyloxazol-5(4H)-one as a new scaffold for selective reversible MAGL inhibitors. (2nd January 2016) Authors: Granchi, Carlotta; Rizzolio, Flavio; Bordoni, Vittorio; Caligiuri, Isabella; Manera, Clementina; Macchia, Marco; Minutolo, Filippo; Martinelli, Adriano; Giordano, Antonio; Tuccinardi, Tiziano Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 31:Number 1(2016:Feb.) Page Start: 137 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. A Single‐Stranded DNA‐Encoded Chemical Library Based on a Stereoisomeric Scaffold Enables Ligand Discovery by Modular Assembly of Building Blocks. Issue 22 (14th October 2020) Authors: Bassi, Gabriele; Favalli, Nicholas; Vuk, Miriam; Catalano, Marco; Martinelli, Adriano; Trenner, Anika; Porro, Antonio; Yang, Su; Tham, Chuin Lean; Moroglu, Mustafa; Yue, Wyatt W.; Conway, Stuart J.; Vogt, Peter K.; Sartori, Alessandro A.; Scheuermann, Jörg; Neri, Dario Journal: Advanced science Issue: Volume 7:Issue 22(2020) Page Start: n/a Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. A Virtual Screening Study for Lactate Dehydrogenase 5 Inhibitors by Using a Pharmacophore‐based Approach. Issue 8 (15th June 2016) Authors: Tuccinardi, Tiziano; Poli, Giulio; Corchia, Isacco; Granchi, Carlotta; Lapillo, Margherita; Macchia, Marco; Minutolo, Filippo; Ortore, Gabriella; Martinelli, Adriano Journal: Molecular informatics Issue: Volume 35:Issue 8/9(2016) Page Start: 434 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Development of a cheminformatics platform for selectivity analyses of carbonic anhydrase inhibitors. (1st January 2020) Authors: Poli, Giulio; Galati, Salvatore; Martinelli, Adriano; Supuran, Claudiu T.; Tuccinardi, Tiziano Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 35:Number 1(2020) Page Start: 365 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Development of terphenyl-2-methyloxazol-5(4H)-one derivatives as selective reversible MAGL inhibitors. (1st January 2017) Authors: Granchi, Carlotta; Caligiuri, Isabella; Bertelli, Eleonora; Poli, Giulio; Rizzolio, Flavio; Macchia, Marco; Martinelli, Adriano; Minutolo, Filippo; Tuccinardi, Tiziano Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 32:Number 1(2017) Page Start: 1240 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Dual Targeting of the Warburg Effect with a Glucose‐Conjugated Lactate Dehydrogenase Inhibitor. Issue 17 (31st October 2013) Authors: Calvaresi, Emilia C.; Granchi, Carlotta; Tuccinardi, Tiziano; Di Bussolo, Valeria; Huigens, Robert W.; Lee, Hyang Yeon; Palchaudhuri, Rahul; Macchia, Marco; Martinelli, Adriano; Minutolo, Filippo; Hergenrother, Paul J. Journal: Chembiochem Issue: Volume 14:Issue 17(2013) Page Start: 2263 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Identification of a new STAT3 dimerization inhibitor through a pharmacophore-based virtual screening approach. (1st November 2016) Authors: Poli, Giulio; Gelain, Arianna; Porta, Federica; Asai, Akira; Martinelli, Adriano; Tuccinardi, Tiziano Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 31:Number 6(2016:Dec.) Page Start: 1011 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Identification of Transthyretin Fibril Formation Inhibitors Using Structure‐Based Virtual Screening. (11th May 2017) Authors: Ortore, Gabriella; Martinelli, Adriano Journal: ChemMedChem Issue: Volume 12:Number 16(2017) Page Start: 1327 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Phenylpropanoids and flavonoids from Phlomis kurdica as inhibitors of human lactate dehydrogenase. (August 2015) Authors: Bader, Ammar; Tuccinardi, Tiziano; Granchi, Carlotta; Martinelli, Adriano; Macchia, Marco; Minutolo, Filippo; De Tommasi, Nunziatina; Braca, Alessandra Journal: Phytochemistry Issue: Volume 116(2015:Aug.) Page Start: 262 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. Phenylpropanoids and flavonoids from Phlomis kurdica as inhibitors of human lactate dehydrogenase. (August 2015) Authors: Bader, Ammar; Tuccinardi, Tiziano; Granchi, Carlotta; Martinelli, Adriano; Macchia, Marco; Minutolo, Filippo; De Tommasi, Nunziatina; Braca, Alessandra Journal: Phytochemistry Issue: Volume 116(2015:Aug.) Page Start: 262 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗