1. Mechanism-based inhibitors of SIRT2: structure–activity relationship, X-ray structures, target engagement, regulation of α-tubulin acetylation and inhibition of breast cancer cell migration. Issue 2 (14th January 2021) Authors: Nielsen, Alexander L.; Rajabi, Nima; Kudo, Norio; Lundø, Kathrine; Moreno-Yruela, Carlos; Bæk, Michael; Fontenas, Martin; Lucidi, Alessia; Madsen, Andreas S.; Yoshida, Minoru; Olsen, Christian A. Journal: RSC chemical biology Issue: Volume 2:Issue 2(2021) Page Start: 612 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Pyrrole- and indole-containing tranylcypromine derivatives as novel lysine-specific demethylase 1 inhibitors active on cancer cells1. Issue 4 (10th April 2015) Authors: Rodriguez, Veronica; Valente, Sergio; Rovida, Stefano; Rotili, Dante; Stazi, Giulia; Lucidi, Alessia; Ciossani, Giuseppe; Mattevi, Andrea; Botrugno, Oronza A.; Dessanti, Paola; Mercurio, Ciro; Vianello, Paola; Minucci, Saverio; Varasi, Mario; Mai, Antonello Journal: MedChemComm Issue: Volume 6:Issue 4(2015:Apr.) Page Start: 665 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Synthesis and characterisation of a new benzamide-containing nitrobenzoxadiazole as a GSTP1-1 inhibitor endowed with high stability to metabolic hydrolysis. (1st January 2019) Authors: Di Paolo, Veronica; Fulci, Chiara; Rotili, Dante; Sciarretta, Francesca; Lucidi, Alessia; Morozzo della Rocca, Blasco; De Luca, Anastasia; Rosato, Antonio; Quintieri, Luigi; Caccuri, Anna Maria Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 34:Number 1(2019) Page Start: 1131 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗