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Author/Creator Leurs, Rob

1. Photoswitching the Efficacy of a Small‐Molecule Ligand for a Peptidergic GPCR: from Antagonism to Agonism. Issue 36 (6th August 2018)

Authors:
Gómez‐Santacana, Xavier; de Munnik, Sabrina M.; Vijayachandran, Prashanna; Da Costa Pereira, Daniel; Bebelman, Jan Paul M.; de Esch, Iwan J. P.; Vischer, Henry F.; Wijtmans, Maikel; Leurs, Rob
Journal:
Angewandte Chemie international edition
Issue:
Volume 57:Issue 36(2018)
Page Start:
11608
Record Type:
Journal Article
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2. Photoswitching the Efficacy of a Small‐Molecule Ligand for a Peptidergic GPCR: from Antagonism to Agonism. (6th August 2018)

Authors:
Gómez‐Santacana, Xavier; de Munnik, Sabrina M.; Vijayachandran, Prashanna; Da Costa Pereira, Daniel; Bebelman, Jan Paul M.; de Esch, Iwan J. P.; Vischer, Henry F.; Wijtmans, Maikel; Leurs, Rob
Journal:
Angewandte Chemie
Issue:
Volume 130:Number 36(2018)
Page Start:
11782
Record Type:
Journal Article
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3. Identification of Phenylpyrazolone Dimers as a New Class of Anti‐Trypanosoma cruzi Agents. (23rd August 2019)

Authors:
Sijm, Maarten; Siciliano de Araújo, Julianna; Ramos Llorca, Alba; Orrling, Kristina; Stiny, Lydia; Matheeussen, An; Maes, Louis; de Esch, Iwan J. P.; de Nazaré Correia Soeiro, Maria; Sterk, Geert Jan; Leurs, Rob
Journal:
ChemMedChem
Issue:
Volume 14:Number 18(2019)
Page Start:
1662
Record Type:
Journal Article
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4. Histamine receptors in GtoPdb v.2021.3. (2021)

Authors:
Chazot, Paul; Cowart, Marlon; Fukui, Hiroyuki; Ganellin, C. Robin; Gutzmer, Ralf; Haas, Helmut L.; Hill, Stephen J.; Hills, Rebecca; Leurs, Rob; Levi, Roberto; Liu, Steve; Panula, Pertti; Schunack, Walter; Schwartz, Jean-Charles; Seifert, Roland; Shankley, Nigel P.; Stark, Holger; Thurmond, Robin...
Journal:
IUPHAR/BPS guide to pharmacology CITE
Issue:
Number 3(2021)
Page Start:
Record Type:
Journal Article
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6. Kinetics for Drug Discovery: an industry-driven effort to target drug residence time. Issue 6 (June 2017)

Authors:
Schuetz, Doris A.; de Witte, Wilhelmus Egbertus Arnout; Wong, Yin Cheong; Knasmueller, Bernhard; Richter, Lars; Kokh, Daria B.; Sadiq, S. Kashif; Bosma, Reggie; Nederpelt, Indira; Heitman, Laura H.; Segala, Elena; Amaral, Marta; Guo, Dong; Andres, Dorothee; Georgi, Victoria; Stoddart, Leigh A.; H...
Journal:
Drug discovery today
Issue:
Volume 22:Issue 6(2017)
Page Start:
896
Record Type:
Journal Article
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7. Alkynamide phthalazinones as a new class of TbrPDEB1 inhibitors. Issue 18 (15th September 2019)

Authors:
de Heuvel, Erik; Singh, Abhimanyu K.; Edink, Ewald; van der Meer, Tiffany; van der Woude, Melanie; Sadek, Payman; Krell-Jørgensen, Mikkel P.; van den Bergh, Toine; Veerman, Johan; Caljon, Guy; Kalejaiye, Titilola D.; Wijtmans, Maikel; Maes, Louis; de Koning, Harry P.; Jan Sterk, Geert; Siderius, ...
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 27:Issue 18(2019)
Page Start:
3998
Record Type:
Journal Article
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8. Alkynamide phthalazinones as a new class of TbrPDEB1 inhibitors (Part 2). Issue 18 (15th September 2019)

Authors:
de Heuvel, Erik; Singh, Abhimanyu K.; Boronat, Pierre; Kooistra, Albert J.; van der Meer, Tiffany; Sadek, Payman; Blaazer, Antoni R.; Shaner, Nathan C.; Bindels, Daphne S.; Caljon, Guy; Maes, Louis; Sterk, Geert Jan; Siderius, Marco; Oberholzer, Michael; de Esch, Iwan J.P.; Brown, David G.; Leurs...
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 27:Issue 18(2019)
Page Start:
4013
Record Type:
Journal Article
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9. A Photoswitchable Agonist for the Histamine H3 Receptor, a Prototypic Family A G‐Protein‐Coupled Receptor. Issue 14 (27th February 2019)

Authors:
Hauwert, Niels J.; Mocking, Tamara A. M.; Da Costa Pereira, Daniel; Lion, Ken; Huppelschoten, Yara; Vischer, Henry F.; De Esch, Iwan J. P.; Wijtmans, Maikel; Leurs, Rob
Journal:
Angewandte Chemie international edition
Issue:
Volume 58:Issue 14(2019)
Page Start:
4531
Record Type:
Journal Article
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10. A Photoswitchable Agonist for the Histamine H3 Receptor, a Prototypic Family A G‐Protein‐Coupled Receptor. (27th February 2019)

Authors:
Hauwert, Niels J.; Mocking, Tamara A. M.; Da Costa Pereira, Daniel; Lion, Ken; Huppelschoten, Yara; Vischer, Henry F.; De Esch, Iwan J. P.; Wijtmans, Maikel; Leurs, Rob
Journal:
Angewandte Chemie
Issue:
Volume 131:Number 14(2019)
Page Start:
4579
Record Type:
Journal Article
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