1. ASP5878, a selective FGFR inhibitor, to treat FGFR3‐dependent urothelial cancer with or without chemoresistance. Issue 2 (February 2017) Authors: Kikuchi, Aya; Suzuki, Tomoyuki; Nakazawa, Taisuke; Iizuka, Masateru; Nakayama, Ayako; Ozawa, Tohru; Kameda, Minoru; Shindoh, Nobuaki; Terasaka, Tadashi; Hirano, Masaaki; Kuromitsu, Sadao Journal: Cancer science Issue: Volume 108:Issue 2(2017) Page Start: 236 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Discovery of ASP5878: Synthesis and structure–activity relationships of pyrimidine derivatives as pan-FGFRs inhibitors with improved metabolic stability and suppressed hERG channel inhibitory activity. (1st April 2022) Authors: Kuriwaki, Ikumi; Kameda, Minoru; Iikubo, Kazuhiko; Hisamichi, Hiroyuki; Kawamoto, Yuichiro; Kikuchi, Shigetoshi; Moritomo, Hiroyuki; Terasaka, Tadashi; Iwai, Yoshinori; Noda, Atsushi; Tomiyama, Hiroshi; Kikuchi, Aya; Hirano, Masaaki Journal: Bioorganic & medicinal chemistry Issue: Volume 59(2022) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Structure-based drug design of 1, 3, 5-triazine and pyrimidine derivatives as novel FGFR3 inhibitors with high selectivity over VEGFR2. Issue 10 (15th May 2020) Authors: Kuriwaki, Ikumi; Kameda, Minoru; Hisamichi, Hiroyuki; Kikuchi, Shigetoshi; Iikubo, Kazuhiko; Kawamoto, Yuichiro; Moritomo, Hiroyuki; Kondoh, Yutaka; Amano, Yasushi; Tateishi, Yukihiro; Echizen, Yuka; Iwai, Yoshinori; Noda, Atsushi; Tomiyama, Hiroshi; Suzuki, Tomoyuki; Hirano, Masaaki Journal: Bioorganic & medicinal chemistry Issue: Volume 28:Issue 10(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Synthesis and structure-activity relationships of pyrimidine derivatives as potent and orally active FGFR3 inhibitors with both increased systemic exposure and enhanced in vitro potency. (1st March 2021) Authors: Kuriwaki, Ikumi; Kameda, Minoru; Iikubo, Kazuhiko; Hisamichi, Hiroyuki; Kawamoto, Yuichiro; Kikuchi, Shigetoshi; Moritomo, Hiroyuki; Kondoh, Yutaka; Terasaka, Tadashi; Amano, Yasushi; Tateishi, Yukihiro; Echizen, Yuka; Iwai, Yoshinori; Noda, Atsushi; Tomiyama, Hiroshi; Nakazawa, Taisuke; Hirano, ... Journal: Bioorganic & medicinal chemistry Issue: Volume 33(2021) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗