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Author/Creator Kameda, Minoru

1. ASP5878, a selective FGFR inhibitor, to treat FGFR3‐dependent urothelial cancer with or without chemoresistance. Issue 2 (February 2017)

Authors:
Kikuchi, Aya; Suzuki, Tomoyuki; Nakazawa, Taisuke; Iizuka, Masateru; Nakayama, Ayako; Ozawa, Tohru; Kameda, Minoru; Shindoh, Nobuaki; Terasaka, Tadashi; Hirano, Masaaki; Kuromitsu, Sadao
Journal:
Cancer science
Issue:
Volume 108:Issue 2(2017)
Page Start:
236
Record Type:
Journal Article
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2. Discovery of ASP5878: Synthesis and structure–activity relationships of pyrimidine derivatives as pan-FGFRs inhibitors with improved metabolic stability and suppressed hERG channel inhibitory activity. (1st April 2022)

Authors:
Kuriwaki, Ikumi; Kameda, Minoru; Iikubo, Kazuhiko; Hisamichi, Hiroyuki; Kawamoto, Yuichiro; Kikuchi, Shigetoshi; Moritomo, Hiroyuki; Terasaka, Tadashi; Iwai, Yoshinori; Noda, Atsushi; Tomiyama, Hiroshi; Kikuchi, Aya; Hirano, Masaaki
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 59(2022)
Page Start:
Record Type:
Journal Article
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3. Structure-based drug design of 1, 3, 5-triazine and pyrimidine derivatives as novel FGFR3 inhibitors with high selectivity over VEGFR2. Issue 10 (15th May 2020)

Authors:
Kuriwaki, Ikumi; Kameda, Minoru; Hisamichi, Hiroyuki; Kikuchi, Shigetoshi; Iikubo, Kazuhiko; Kawamoto, Yuichiro; Moritomo, Hiroyuki; Kondoh, Yutaka; Amano, Yasushi; Tateishi, Yukihiro; Echizen, Yuka; Iwai, Yoshinori; Noda, Atsushi; Tomiyama, Hiroshi; Suzuki, Tomoyuki; Hirano, Masaaki
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 28:Issue 10(2020)
Page Start:
Record Type:
Journal Article
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4. Synthesis and structure-activity relationships of pyrimidine derivatives as potent and orally active FGFR3 inhibitors with both increased systemic exposure and enhanced in vitro potency. (1st March 2021)

Authors:
Kuriwaki, Ikumi; Kameda, Minoru; Iikubo, Kazuhiko; Hisamichi, Hiroyuki; Kawamoto, Yuichiro; Kikuchi, Shigetoshi; Moritomo, Hiroyuki; Kondoh, Yutaka; Terasaka, Tadashi; Amano, Yasushi; Tateishi, Yukihiro; Echizen, Yuka; Iwai, Yoshinori; Noda, Atsushi; Tomiyama, Hiroshi; Nakazawa, Taisuke; Hirano, ...
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 33(2021)
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Record Type:
Journal Article
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