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Author/Creator Hopkins, Corey R.

3. Design, synthesis and characterization of novel N-heterocyclic-1-benzyl-1H-benzo[d]imidazole-2-amines as selective TRPC5 inhibitors leading to the identification of the selective compound, AC1903. Issue 2 (15th January 2019)

Authors:
Sharma, Swagat H.; Pablo, Juan Lorenzo; Montesinos, Monica Suarez; Greka, Anna; Hopkins, Corey R.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 29:Issue 2(2019)
Page Start:
155
Record Type:
Journal Article
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4. Discovery and Characterization of 2‐(Cyclopropanesulfonamido)‐N‐(2‐ethoxyphenyl)benzamide, ML382: a Potent and Selective Positive Allosteric Modulator of MrgX1. Issue 1 (10th September 2014)

Authors:
Wen, Wandong; Wang, Yan; Li, Zhe; Tseng, Pang‐Yen; McManus, Owen B.; Wu, Meng; Li, Min; Lindsley, Craig W.; Dong, Xinzhong; Hopkins, Corey R.
Journal:
ChemMedChem
Issue:
Volume 10:Issue 1(2015:Jan.)
Page Start:
57
Record Type:
Journal Article
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5. Discovery and characterization of a novel series of N-phenylsulfonyl-1H-pyrrole picolinamides as positive allosteric modulators of the metabotropic glutamate receptor 4 (mGlu4). Issue 13 (1st July 2016)

Authors:
Gogliotti, Rocco D.; Blobaum, Anna L.; Morrison, Ryan M.; Daniels, J. Scott; Salovich, James M.; Cheung, Yiu-Yin; Rodriguez, Alice L.; Loch, Matthew T.; Conn, P. Jeffrey; Lindsley, Craig W.; Niswender, Colleen M.; Hopkins, Corey R.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 13(2016)
Page Start:
2984
Record Type:
Journal Article
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7. Discovery and characterization of N-(1, 3-dialkyl-1H-indazol-6-yl)-1H-pyrazolo[4, 3-b]pyridin-3-amine scaffold as mGlu4 positive allosteric modulators that mitigate CYP1A2 induction liability. Issue 15 (15th August 2018)

Authors:
Engers, Darren W.; Bollinger, Sean R.; Engers, Julie L.; Panarese, Joseph D.; Breiner, Megan M.; Gregro, Alison; Blobaum, Anna L.; Bronson, Joanne J.; Wu, Yong-Jin; Macor, John E.; Rodriguez, Alice L.; Zamorano, Rocio; Conn, P. Jeffrey; Lindsley, Craig W.; Niswender, Colleen M.; Hopkins, Corey R.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 28:Issue 15(2018)
Page Start:
2641
Record Type:
Journal Article
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8. Discovery and optimization of a novel series of highly CNS penetrant M4 PAMs based on a 5, 6-dimethyl-4-(piperidin-1-yl)thieno[2, 3-d]pyrimidine core. Issue 13 (1st July 2016)

Authors:
Wood, Michael R.; Noetzel, Meredith J.; Engers, Julie L.; Bollinger, Katrina A.; Melancon, Bruce J.; Tarr, James C.; Han, Changho; West, Mary; Gregro, Alison R.; Lamsal, Atin; Chang, Sichen; Ajmera, Sonia; Smith, Emery; Chase, Peter; Hodder, Peter S.; Bubser, Michael; Jones, Carrie K.; Hopkins, C...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 13(2016)
Page Start:
3029
Record Type:
Journal Article
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9. Discovery of 3-aminopicolinamides as metabotropic glutamate receptor subtype 4 (mGlu4) positive allosteric modulator warheads engendering CNS exposure and in vivo efficacy. Issue 12 (15th June 2016)

Authors:
Gogliotti, Rocco D.; Engers, Darren W.; Garcia-Barrantes, Pedro M.; Panarese, Joseph D.; Gentry, Patrick R.; Blobaum, Anna L.; Morrison, Ryan D.; Daniels, J. Scott; Thompson, Analisa D.; Jones, Carrie K.; Conn, P. Jeffrey; Niswender, Colleen M.; Lindsley, Craig W.; Hopkins, Corey R.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 12(2016)
Page Start:
2915
Record Type:
Journal Article
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10. Discovery, characterization and biological evaluation of a novel (R)-4, 4-difluoropiperidine scaffold as dopamine receptor 4 (D4R) antagonists. Issue 23 (1st December 2016)

Authors:
Jeffries, Daniel E.; Witt, Jonathan O.; McCollum, Andrea L.; Temple, Kayla J.; Hurtado, Miguel A.; Harp, Joel M.; Blobaum, Anna L.; Lindsley, Craig W.; Hopkins, Corey R.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 23(2016)
Page Start:
5757
Record Type:
Journal Article
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