1. Activity cliff for 7-substituted pyrrolo-pyrimidine inhibitors of HCK explained in terms of predicted basicity of the amine nitrogen. Issue 16 (15th August 2017) Authors: Yuki, Hitomi; Kikuzato, Ko; Koda, Yasuko; Mikuni, Junko; Tomabechi, Yuri; Kukimoto-Niino, Mutsuko; Tanaka, Akiko; Shirai, Fumiyuki; Shirouzu, Mikako; Koyama, Hiroo; Honma, Teruki Journal: Bioorganic & medicinal chemistry Issue: Volume 25:Issue 16(2017) Page Start: 4259 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Characterization of crystal water molecules in a high-affinity inhibitor and hematopoietic prostaglandin D synthase complex by interaction energy studies. Issue 16 (1st September 2018) Authors: Takaya, Daisuke; Inaka, Koji; Omura, Akifumi; Takenuki, Kenji; Kawanishi, Masashi; Yabuki, Yukako; Nakagawa, Yukari; Tsuganezawa, Keiko; Ogawa, Naoko; Watanabe, Chiduru; Honma, Teruki; Aritake, Kosuke; Urade, Yoshihiro; Shirouzu, Mikako; Tanaka, Akiko Journal: Bioorganic & medicinal chemistry Issue: Volume 26:Issue 16(2018) Page Start: 4726 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Design and synthesis of potent substrate-based inhibitors of the Trypanosoma cruzi dihydroorotate dehydrogenase. Issue 4 (15th February 2017) Authors: Inaoka, Daniel Ken; Iida, Maiko; Hashimoto, Satoshi; Tabuchi, Toshiyuki; Kuranaga, Takefumi; Balogun, Emmanuel Oluwadare; Honma, Teruki; Tanaka, Akiko; Harada, Shigeharu; Nara, Takeshi; Kita, Kiyoshi; Inoue, Masayuki Journal: Bioorganic & medicinal chemistry Issue: Volume 25:Issue 4(2017) Page Start: 1465 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Interruption of Vif/Elongin C interaction: In silico and experimental elucidation of the underlying molecular mechanism of benzimidazole-based APOBEC3G stabilizers. Issue 8 (15th April 2020) Authors: Radwan, Mohamed O.; Takaya, Daisuke; Koga, Ryoko; Iwamaru, Kana; Tateishi, Hiroshi; Ali, Taha F.S.; Takaori-Kondo, Akifumi; Otsuka, Masami; Honma, Teruki; Fujita, Mikako Journal: Bioorganic & medicinal chemistry Issue: Volume 28:Issue 8(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. New antimalarials identified by a cell-based phenotypic approach: Structure–activity relationships of 2, 3, 4, 9-tetrahydro-1H-β-carboline derivatives possessing a 2-((coumarin-5-yl)oxy)alkanoyl moiety. (15th July 2022) Authors: Cho, Nobuo; Kikuzato, Ko; Futamura, Yushi; Shimizu, Takeshi; Hayase, Hiroki; Kamisaka, Kikuko; Takaya, Daisuke; Yuki, Hitomi; Honma, Teruki; Niikura, Mamoru; Kobayashi, Fumie; Watanabe, Nobumoto; Osada, Hiroyuki; Koyama, Hiroo Journal: Bioorganic & medicinal chemistry Issue: Volume 66(2022) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. New SIRT2 inhibitors: Histidine-based bleomycin spin-off. Issue 9 (1st May 2019) Authors: Ali, Taha F.S.; Ciftci, Halil I.; Radwan, Mohamed O.; Koga, Ryoko; Ohsugi, Takeo; Okiyama, Yoshio; Honma, Teruki; Nakata, Akiko; Ito, Akihiro; Yoshida, Minoru; Fujita, Mikako; Otsuka, Masami Journal: Bioorganic & medicinal chemistry Issue: Volume 27:Issue 9(2019) Page Start: 1767 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗