1. A public–private partnership to enrich the development of in silico predictive models for pharmacokinetic and cardiotoxic properties. Issue 5 (May 2021) Authors: Komura, Hiroshi; Watanabe, Reiko; Kawashima, Hitoshi; Ohashi, Rikiya; Kuroda, Masataka; Sato, Tomohiro; Honma, Teruki; Mizuguchi, Kenji Journal: Drug discovery today Issue: Volume 26:Issue 5(2021) Page Start: 1275 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Activity cliff for 7-substituted pyrrolo-pyrimidine inhibitors of HCK explained in terms of predicted basicity of the amine nitrogen. Issue 16 (15th August 2017) Authors: Yuki, Hitomi; Kikuzato, Ko; Koda, Yasuko; Mikuni, Junko; Tomabechi, Yuri; Kukimoto-Niino, Mutsuko; Tanaka, Akiko; Shirai, Fumiyuki; Shirouzu, Mikako; Koyama, Hiroo; Honma, Teruki Journal: Bioorganic & medicinal chemistry Issue: Volume 25:Issue 16(2017) Page Start: 4259 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Alantolactone is a natural product that potently inhibits YAP1/TAZ through promotion of reactive oxygen species accumulation. Issue 10 (6th August 2021) Authors: Nakatani, Keisuke; Maehama, Tomohiko; Nishio, Miki; Otani, Junji; Yamaguchi, Keiko; Fukumoto, Miki; Hikasa, Hiroki; Hagiwara, Shinji; Nishina, Hiroshi; Mak, Tak Wah; Honma, Teruki; Kondoh, Yasumitsu; Osada, Hiroyuki; Yoshida, Minoru; Suzuki, Akira Journal: Cancer science Issue: Volume 112:Issue 10(2021) Page Start: 4303 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Anthocyanin 5, 3′-aromatic acyltransferase from Gentiana triflora, a structural insight into biosynthesis of a blue anthocyanin. (June 2021) Authors: Murayama, Kazutaka; Kato-Murayama, Miyuki; Sato, Tomohiro; Hosaka, Toshiaki; Ishiguro, Kanako; Mizuno, Takayuki; Kitao, Kazunori; Honma, Teruki; Yokoyama, Shigeyuki; Tanaka, Yoshikazu; Shirouzu, Mikako Journal: Phytochemistry Issue: Volume 186(2021) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Characterization of crystal water molecules in a high-affinity inhibitor and hematopoietic prostaglandin D synthase complex by interaction energy studies. Issue 16 (1st September 2018) Authors: Takaya, Daisuke; Inaka, Koji; Omura, Akifumi; Takenuki, Kenji; Kawanishi, Masashi; Yabuki, Yukako; Nakagawa, Yukari; Tsuganezawa, Keiko; Ogawa, Naoko; Watanabe, Chiduru; Honma, Teruki; Aritake, Kosuke; Urade, Yoshihiro; Shirouzu, Mikako; Tanaka, Akiko Journal: Bioorganic & medicinal chemistry Issue: Volume 26:Issue 16(2018) Page Start: 4726 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Design and synthesis of potent substrate-based inhibitors of the Trypanosoma cruzi dihydroorotate dehydrogenase. Issue 4 (15th February 2017) Authors: Inaoka, Daniel Ken; Iida, Maiko; Hashimoto, Satoshi; Tabuchi, Toshiyuki; Kuranaga, Takefumi; Balogun, Emmanuel Oluwadare; Honma, Teruki; Tanaka, Akiko; Harada, Shigeharu; Nara, Takeshi; Kita, Kiyoshi; Inoue, Masayuki Journal: Bioorganic & medicinal chemistry Issue: Volume 25:Issue 4(2017) Page Start: 1465 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Discovery of trypanocidal coumarins with dual inhibition of both the glycerol kinase and alternative oxidase of Trypanosoma brucei brucei. Issue 11 (16th September 2019) Authors: Balogun, Emmanuel Oluwadare; Inaoka, Daniel Ken; Shiba, Tomoo; Tsuge, Chiaki; May, Benjamin; Sato, Tomohiro; Kido, Yasutoshi; Nara, Takeshi; Aoki, Takashi; Honma, Teruki; Tanaka, Akiko; Inoue, Masayuki; Matsuoka, Shigeru; Michels, Paul A. M.; Watanabe, Yoh‐Ichi; Moore, Anthony L.; Harada, Shigeha... Journal: FASEB journal Issue: Volume 33:Issue 11(2019) Page Start: 13002 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Identification of pyrrolo[2, 3-d]pyrimidines as potent HCK and FLT3-ITD dual inhibitors. Issue 22 (15th November 2017) Authors: Koda, Yasuko; Kikuzato, Ko; Mikuni, Junko; Tanaka, Akiko; Yuki, Hitomi; Honma, Teruki; Tomabechi, Yuri; Kukimoto-Niino, Mutsuko; Shirouzu, Mikako; Shirai, Fumiyuki; Koyama, Hiroo Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 22(2017) Page Start: 4994 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Interruption of Vif/Elongin C interaction: In silico and experimental elucidation of the underlying molecular mechanism of benzimidazole-based APOBEC3G stabilizers. Issue 8 (15th April 2020) Authors: Radwan, Mohamed O.; Takaya, Daisuke; Koga, Ryoko; Iwamaru, Kana; Tateishi, Hiroshi; Ali, Taha F.S.; Takaori-Kondo, Akifumi; Otsuka, Masami; Honma, Teruki; Fujita, Mikako Journal: Bioorganic & medicinal chemistry Issue: Volume 28:Issue 8(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. Molecular basis for the reverse reaction of African human trypanosomes glycerol kinase. Issue 6 (4th November 2014) Authors: Balogun, Emmanuel Oluwadare; Inaoka, Daniel Ken; Shiba, Tomoo; Kido, Yasutoshi; Tsuge, Chiaki; Nara, Takeshi; Aoki, Takashi; Honma, Teruki; Tanaka, Akiko; Inoue, Masayuki; Matsuoka, Shigeru; Michels, Paul A. M.; Kita, Kiyoshi; Harada, Shigeharu Journal: Molecular microbiology Issue: Volume 94:Issue 6(2014) Page Start: 1315 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗