1. 8-Substituted 1, 3-dimethyltetrahydropyrazino[2, 1-f]purinediones: Water-soluble adenosine receptor antagonists and monoamine oxidase B inhibitors. Issue 21 (1st November 2016) Authors: Brunschweiger, Andreas; Koch, Pierre; Schlenk, Miriam; Rafehi, Muhammad; Radjainia, Hamid; Küppers, Petra; Hinz, Sonja; Pineda, Felipe; Wiese, Michael; Hockemeyer, Jörg; Heer, Jag; Denonne, Frédéric; Müller, Christa E. Journal: Bioorganic & medicinal chemistry Issue: Volume 24:Issue 21(2016) Page Start: 5462 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. 8‐Benzyltetrahydropyrazino[2, 1‐f]purinediones: Water‐Soluble Tricyclic Xanthine Derivatives as Multitarget Drugs for Neurodegenerative Diseases. Issue 8 (9th May 2014) Authors: Brunschweiger, Andreas; Koch, Pierre; Schlenk, Miriam; Pineda, Felipe; Küppers, Petra; Hinz, Sonja; Köse, Meryem; Ullrich, Stefan; Hockemeyer, Jörg; Wiese, Michael; Heer, Jag; Müller, Christa E. Journal: ChemMedChem Issue: Volume 9:Issue 8(2014:Aug.) Page Start: 1704 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Back Cover: Discovery of a PCAF Bromodomain Chemical Probe (Angew. Chem. Int. Ed. 3/2017). Issue 3 (23rd December 2016) Authors: Moustakim, Moses; Clark, Peter G. K.; Trulli, Laura; Fuentes de Arriba, Angel L.; Ehebauer, Matthias T.; Chaikuad, Apirat; Murphy, Emma J.; Mendez‐Johnson, Jacqui; Daniels, Danette; Hou, Chun‐Feng D.; Lin, Yu‐Hui; Walker, John R.; Hui, Raymond; Yang, Hongbing; Dorrell, Lucy; Rogers, Catherine M.;... Journal: Angewandte Chemie international edition Issue: Volume 56:Issue 3(2017) Page Start: 908 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Discovery of a novel allosteric inhibitor scaffold for polyadenosine-diphosphate-ribose polymerase 14 (PARP14) macrodomain 2. Issue 11 (15th July 2018) Authors: Moustakim, Moses; Riedel, Kerstin; Schuller, Marion; Gehring, Andrè P.; Monteiro, Octovia P.; Martin, Sarah P.; Fedorov, Oleg; Heer, Jag; Dixon, Darren J.; Elkins, Jonathan M.; Knapp, Stefan; Bracher, Franz; Brennan, Paul E. Journal: Bioorganic & medicinal chemistry Issue: Volume 26:Issue 11(2018) Page Start: 2965 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Discovery of a PCAF Bromodomain Chemical Probe. (14th December 2016) Authors: Moustakim, Moses; Clark, Peter G. K.; Trulli, Laura; Fuentes de Arriba, Angel L.; Ehebauer, Matthias T.; Chaikuad, Apirat; Murphy, Emma J.; Mendez‐Johnson, Jacqui; Daniels, Danette; Hou, Chun‐Feng D.; Lin, Yu‐Hui; Walker, John R.; Hui, Raymond; Yang, Hongbing; Dorrell, Lucy; Rogers, Catherine M.;... Journal: Angewandte Chemie Issue: Volume 129:Number 3(2017) Page Start: 845 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Discovery of a PCAF Bromodomain Chemical Probe. Issue 3 (14th December 2016) Authors: Moustakim, Moses; Clark, Peter G. K.; Trulli, Laura; Fuentes de Arriba, Angel L.; Ehebauer, Matthias T.; Chaikuad, Apirat; Murphy, Emma J.; Mendez‐Johnson, Jacqui; Daniels, Danette; Hou, Chun‐Feng D.; Lin, Yu‐Hui; Walker, John R.; Hui, Raymond; Yang, Hongbing; Dorrell, Lucy; Rogers, Catherine M.;... Journal: Angewandte Chemie international edition Issue: Volume 56:Issue 3(2017) Page Start: 827 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Discovery of an MLLT1/3 YEATS Domain Chemical Probe. Issue 50 (16th November 2018) Authors: Moustakim, Moses; Christott, Thomas; Monteiro, Octovia P.; Bennett, James; Giroud, Charline; Ward, Jennifer; Rogers, Catherine M.; Smith, Paul; Panagakou, Ioanna; Díaz‐Sáez, Laura; Felce, Suet Ling; Gamble, Vicki; Gileadi, Carina; Halidi, Nadia; Heidenreich, David; Chaikuad, Apirat; Knapp, Stefan... Journal: Angewandte Chemie international edition Issue: Volume 57:Issue 50(2018) Page Start: 16302 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Entdeckung einer chemischen Sonde für MLLT1/3‐YEATS‐Domänen. (16th November 2018) Authors: Moustakim, Moses; Christott, Thomas; Monteiro, Octovia P.; Bennett, James; Giroud, Charline; Ward, Jennifer; Rogers, Catherine M.; Smith, Paul; Panagakou, Ioanna; Díaz‐Sáez, Laura; Felce, Suet Ling; Gamble, Vicki; Gileadi, Carina; Halidi, Nadia; Heidenreich, David; Chaikuad, Apirat; Knapp, Stefan... Journal: Angewandte Chemie Issue: Volume 130:Number 50(2018) Page Start: 16540 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Rücktitelbild: Discovery of a PCAF Bromodomain Chemical Probe (Angew. Chem. 3/2017). (23rd December 2016) Authors: Moustakim, Moses; Clark, Peter G. K.; Trulli, Laura; Fuentes de Arriba, Angel L.; Ehebauer, Matthias T.; Chaikuad, Apirat; Murphy, Emma J.; Mendez‐Johnson, Jacqui; Daniels, Danette; Hou, Chun‐Feng D.; Lin, Yu‐Hui; Walker, John R.; Hui, Raymond; Yang, Hongbing; Dorrell, Lucy; Rogers, Catherine M.;... Journal: Angewandte Chemie Issue: Volume 129:Number 3(2017) Page Start: 928 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗