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Author/Creator Haupenthal, Jörg

4. Biophysical Screening of a Focused Library for the Discovery of CYP121 Inhibitors as Novel Antimycobacterials. (26th September 2017)

Authors:
Brengel, Christian; Thomann, Andreas; Schifrin, Alexander; Allegretta, Giuseppe; Kamal, Ahmed A. M.; Haupenthal, Jörg; Schnorr, Isabell; Cho, Sang Hyun; Franzblau, Scott G.; Empting, Martin; Eberhard, Jens; Hartmann, Rolf W.
Journal:
ChemMedChem
Issue:
Volume 12:Number 19(2017)
Page Start:
1616
Record Type:
Journal Article
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5. CYP17A1-independent production of the neurosteroid-derived 5α-pregnan-3β, 6α-diol-20-one in androgen-responsive prostate cancer cell lines under serum starvation and inhibition by Abiraterone. Issue 174 (November 2017)

Authors:
de Mello Martins, Antonio G. Gomes; Allegretta, Giuseppe; Unteregger, Gerhard; Haupenthal, Jörg; Eberhard, Jens; Hoffmann, Michael; van der Zee, Jill A.; Junker, Kerstin; Stöckle, Michael; Müller, Rolf; Hartmann, Rolf W.; Ohlmann, Carsten-H.
Journal:
Journal of steroid biochemistry and molecular biology
Issue:
Issue 174(2017)
Page Start:
183
Record Type:
Journal Article
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6. Discovery of novel drug-like antitubercular hits targeting the MEP pathway enzyme DXPS by strategic application of ligand-based virtual screening. Issue 36 (7th September 2022)

Authors:
Zhu, Di; Johannsen, Sandra; Masini, Tiziana; Simonin, Céline; Haupenthal, Jörg; Illarionov, Boris; Andreas, Anastasia; Awale, Mahendra; Gierse, Robin M.; van der Laan, Tridia; van der Vlag, Ramon; Nasti, Rita; Poizat, Mael; Buhler, Eric; Reiling, Norbert; Müller, Rolf; Fischer, Markus; Reymond, J...
Journal:
Chemical science
Issue:
Volume 13:Issue 36(2022)
Page Start:
10686
Record Type:
Journal Article
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7. Discovery of the First Selective Nanomolar Inhibitors of ERAP2 by Kinetic Target‐Guided Synthesis. (19th August 2022)

Authors:
Camberlein, Virgyl; Fléau, Charlotte; Sierocki, Pierre; Li, Lenong; Gealageas, Ronan; Bosc, Damien; Guillaume, Valentin; Warenghem, Sandrine; Leroux, Florence; Rosell, Melissa; Cheng, Keguang; Medve, Laura; Prigent, Mathilde; Decanter, Myriam; Piveteau, Catherine; Biela, Alexandre; Eveque, Maxime...
Journal:
Angewandte Chemie
Issue:
Volume 134:Number 39(2022)
Page Start:
n/a
Record Type:
Journal Article
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8. Discovery of the First Selective Nanomolar Inhibitors of ERAP2 by Kinetic Target‐Guided Synthesis. Issue 39 (19th August 2022)

Authors:
Camberlein, Virgyl; Fléau, Charlotte; Sierocki, Pierre; Li, Lenong; Gealageas, Ronan; Bosc, Damien; Guillaume, Valentin; Warenghem, Sandrine; Leroux, Florence; Rosell, Melissa; Cheng, Keguang; Medve, Laura; Prigent, Mathilde; Decanter, Myriam; Piveteau, Catherine; Biela, Alexandre; Eveque, Maxime...
Journal:
Angewandte Chemie international edition
Issue:
Volume 61:Issue 39(2022)
Page Start:
n/a
Record Type:
Journal Article
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9. Front Cover: Phosphonate as a Stable Zinc‐Binding Group for "Pathoblocker" Inhibitors of Clostridial Collagenase H (ColH) (ChemMedChem 8/2021). (22nd April 2021)

Authors:
Voos, Katrin; Schönauer, Esther; Alhayek, Alaa; Haupenthal, Jörg; Andreas, Anastasia; Müller, Rolf; Hartmann, Rolf W.; Brandstetter, Hans; Hirsch, Anna K. H.; Ducho, Christian
Journal:
ChemMedChem
Issue:
Volume 16:Number 8(2021)
Page Start:
1198
Record Type:
Journal Article
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10. Hit-optimization using target-directed dynamic combinatorial chemistry: development of inhibitors of the anti-infective target 1-deoxy-d-xylulose-5-phosphate synthase. Issue 22 (6th May 2021)

Authors:
Jumde, Ravindra P.; Guardigni, Melissa; Gierse, Robin M.; Alhayek, Alaa; Zhu, Di; Hamid, Zhoor; Johannsen, Sandra; Elgaher, Walid A. M.; Neusens, Philipp J.; Nehls, Christian; Haupenthal, Jörg; Reiling, Norbert; Hirsch, Anna K. H.
Journal:
Chemical science
Issue:
Volume 12:Issue 22(2021)
Page Start:
7775
Record Type:
Journal Article
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