1. A novel inhibitor stabilizes the inactive conformation of MAPK‐interacting kinase 1. Issue 3 (2nd March 2018) Authors: Matsui, Yumi; Yasumatsu, Isao; Yoshida, Ken-ichi; Iimura, Shin; Ikeno, Yutaka; Nawano, Takako; Fukano, Hajime; Ubukata, Osamu; Hanzawa, Hiroyuki; Tanzawa, Fumie; Isoyama, Takeshi Journal: Acta crystallographica Issue: Volume 74:Issue 3(2018:Mar.) Page Start: 156 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Analysis of fluoroquinolone-resistance using MIC determination and homology modelling of ParC of contemporary Mycoplasma genitalium strains. Issue 3 (March 2022) Authors: Hamasuna, Ryoichi; Hanzawa, Hiroyuki; Moritomo, Ayako; Matsumoto, Masahiro; Aono, Hisami; Tomisaki, Ikko; Akasaka, Takaaki; Fujimoto, Naohiro; Jensen, Jørgen Skov Journal: Journal of infection and chemotherapy Issue: Volume 28:Issue 3(2022) Page Start: 377 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Conformational Plasticity of Cyclic Ras‐Inhibitor Peptides Defines Cell Permeabilization Activity. (16th February 2021) Authors: Takeuchi, Koh; Misaki, Imai; Tokunaga, Yuji; Fujisaki, Miwa; Kamoshida, Hajime; Takizawa, Takeshi; Hanzawa, Hiroyuki; Shimada, Ichio Journal: Angewandte Chemie Issue: Volume 133:Number 12(2021) Page Start: 6641 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Conformational Plasticity of Cyclic Ras‐Inhibitor Peptides Defines Cell Permeabilization Activity. Issue 12 (16th February 2021) Authors: Takeuchi, Koh; Misaki, Imai; Tokunaga, Yuji; Fujisaki, Miwa; Kamoshida, Hajime; Takizawa, Takeshi; Hanzawa, Hiroyuki; Shimada, Ichio Journal: Angewandte Chemie international edition Issue: Volume 60:Issue 12(2021) Page Start: 6567 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Crystal structure of the mineralocorticoid receptor ligand‐binding domain in complex with a potent and selective nonsteroidal blocker, esaxerenone (CS‐3150). Issue 10 (19th February 2020) Authors: Takahashi, Mizuki; Ubukata, Osamu; Homma, Tsuyoshi; Asoh, Yusuke; Honzumi, Masatoshi; Hayashi, Noriyuki; Saito, Keiji; Tsuruoka, Hiroyuki; Aoki, Kazumasa; Hanzawa, Hiroyuki Journal: FEBS letters Issue: Volume 594:Issue 10(2020) Page Start: 1615 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Discovery and structure-guided fragment-linking of 4-(2, 3-dichlorobenzoyl)-1-methyl-pyrrole-2-carboxamide as a pyruvate kinase M2 activator. Issue 13 (1st July 2017) Authors: Matsui, Yumi; Yasumatsu, Isao; Asahi, Takashi; Kitamura, Takahiro; Kanai, Kazuo; Ubukata, Osamu; Hayasaka, Hitoshi; Takaishi, Sachiko; Hanzawa, Hiroyuki; Katakura, Shinichi Journal: Bioorganic & medicinal chemistry Issue: Volume 25:Issue 13(2017) Page Start: 3540 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Discovery and structure-guided optimization of tert-butyl 6-(phenoxymethyl)-3-(trifluoromethyl)benzoates as liver X receptor agonists. Issue 18 (15th September 2015) Authors: Matsui, Yumi; Yamaguchi, Takahiro; Yamazaki, Takanori; Yoshida, Masayuki; Arai, Masami; Terasaka, Naoki; Honzumi, Shoko; Wakabayashi, Kenji; Hayashi, Shinko; Nakai, Daisuke; Hanzawa, Hiroyuki; Tamaki, Kazuhiko Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 18(2015) Page Start: 3914 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Discovery and structure-guided optimization of tert-butyl 6-(phenoxymethyl)-3-(trifluoromethyl)benzoates as liver X receptor agonists. Issue 18 (15th September 2015) Authors: Matsui, Yumi; Yamaguchi, Takahiro; Yamazaki, Takanori; Yoshida, Masayuki; Arai, Masami; Terasaka, Naoki; Honzumi, Shoko; Wakabayashi, Kenji; Hayashi, Shinko; Nakai, Daisuke; Hanzawa, Hiroyuki; Tamaki, Kazuhiko Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 18(2015) Page Start: 3914 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Improvement of Ligand Affinity and Thermodynamic Properties by NMR‐Based Evaluation of Local Dynamics and Surface Complementarity in the Receptor‐Bound State. (20th October 2016) Authors: Mizukoshi, Yumiko; Takeuchi, Koh; Arutaki, Misa; Tokunaga, Yuji; Takizawa, Takeshi; Hanzawa, Hiroyuki; Shimada, Ichio Journal: Angewandte Chemie Issue: Volume 128:Number 47(2016) Page Start: 14826 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. Improvement of Ligand Affinity and Thermodynamic Properties by NMR‐Based Evaluation of Local Dynamics and Surface Complementarity in the Receptor‐Bound State. Issue 47 (20th October 2016) Authors: Mizukoshi, Yumiko; Takeuchi, Koh; Arutaki, Misa; Tokunaga, Yuji; Takizawa, Takeshi; Hanzawa, Hiroyuki; Shimada, Ichio Journal: Angewandte Chemie international edition Issue: Volume 55:Issue 47(2016) Page Start: 14606 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗