11. Discovery of a novel tricyclic 4H-thiazolo[5′, 4′:4, 5]pyrano[2, 3-c]pyridine-2-amino scaffold and its application in a PI3Kα inhibitor with high PI3K isoform selectivity and potent cellular activity. Issue 17 (1st September 2015) Authors: Gerspacher, Marc; Fairhurst, Robin A.; Mah, Robert; Roehn-Carnemolla, Esther; Furet, Pascal; Fritsch, Christine; Guthy, Daniel A. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 17(2015) Page Start: 3582 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
12. Discovery of dihydroisoquinolinone derivatives as novel inhibitors of the p53–MDM2 interaction with a distinct binding mode. Issue 17 (1st September 2015) Authors: Gessier, François; Kallen, Joerg; Jacoby, Edgar; Chène, Patrick; Stachyra-Valat, Thérèse; Ruetz, Stephan; Jeay, Sébastien; Holzer, Philipp; Masuya, Keiichi; Furet, Pascal Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 17(2015) Page Start: 3621 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
13. Front Cover: Structural States of Hdm2 and HdmX: X‐ray Elucidation of Adaptations and Binding Interactions for Different Chemical Compound Classes (ChemMedChem 14/2019). (17th July 2019) Authors: Kallen, Joerg; Izaac, Aude; Chau, Suzanne; Wirth, Emmanuelle; Schoepfer, Joseph; Mah, Robert; Schlapbach, Achim; Stutz, Stefan; Vaupel, Andrea; Guagnano, Vito; Masuya, Keiichi; Stachyra, Therese‐Marie; Salem, Bahaa; Chene, Patrick; Gessier, Francois; Holzer, Philipp; Furet, Pascal Journal: ChemMedChem Issue: Volume 14:Number 14(2019) Page Start: 1304 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
14. Front Cover: The First Class of Small Molecules Potently Disrupting the YAP‐TEAD Interaction by Direct Competition (ChemMedChem 19/2022). (6th October 2022) Authors: Furet, Pascal; Bordas, Vincent; Le Douget, Mickaël; Salem, Bahaa; Mesrouze, Yannick; Imbach‐Weese, Patricia; Sellner, Holger; Voegtle, Markus; Soldermann, Nicolas; Chapeau, Emilie; Wartmann, Markus; Scheufler, Clemens; Fernandez, Cesar; Kallen, Joerg; Guagnano, Vito; Chène, Patrick; Schmelzle, To... Journal: ChemMedChem Issue: Volume 17:Number 19(2022) Page Start: n/a Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
15. Identification and optimisation of 4, 5-dihydrobenzo[1, 2-d:3, 4-d]bisthiazole and 4, 5-dihydrothiazolo[4, 5-h]quinazoline series of selective phosphatidylinositol-3 kinase alpha inhibitors. Issue 17 (1st September 2015) Authors: Fairhurst, Robin A.; Gerspacher, Marc; Imbach-Weese, Patricia; Mah, Robert; Caravatti, Giorgio; Furet, Pascal; Fritsch, Christine; Schnell, Christian; Blanz, Joachim; Blasco, Francesca; Desrayaud, Sandrine; Guthy, Daniel A.; Knapp, Mark; Arz, Dorothee; Wirth, Jasmin; Roehn-Carnemolla, Esther; Luu... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 17(2015) Page Start: 3575 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
16. Identification and optimisation of a 4′, 5-bisthiazole series of selective phosphatidylinositol-3 kinase alpha inhibitors. Issue 17 (1st September 2015) Authors: Fairhurst, Robin A.; Imbach-Weese, Patricia; Gerspacher, Marc; Caravatti, Giorgio; Furet, Pascal; Zoller, Thomas; Fritsch, Christine; Haasen, Dorothea; Trappe, Joerg; Guthy, Daniel A.; Arz, Dorothee; Wirth, Jasmin Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 17(2015) Page Start: 3569 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
17. Identification of a 5-[3-phenyl-(2-cyclic-ether)-methylether]-4-aminopyrrolo[2, 3-d]pyrimidine series of IGF-1R inhibitors. Issue 8 (15th April 2016) Authors: Stauffer, Frédéric; Cowan-Jacob, Sandra W.; Scheufler, Clemens; Furet, Pascal Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 8(2016) Page Start: 2065 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
18. Identification of FAM181A and FAM181B as new interactors with the TEAD transcription factors. (20th November 2019) Authors: Bokhovchuk, Fedir; Mesrouze, Yannick; Delaunay, Clara; Martin, Typhaine; Villard, Frédéric; Meyerhofer, Marco; Fontana, Patrizia; Zimmermann, Catherine; Erdmann, Dirk; Furet, Pascal; Scheufler, Clemens; Schmelzle, Tobias; Chène, Patrick Journal: Protein science Issue: Volume 29:Number 2(2020) Page Start: 509 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
19. In vitro and in vivo characterization of a novel, highly potent p53-MDM2 inhibitor. Issue 20 (1st November 2018) Authors: Vaupel, Andrea; Holzer, Philipp; Ferretti, Stephane; Guagnano, Vito; Kallen, Joerg; Mah, Robert; Masuya, Keiichi; Ruetz, Stephan; Rynn, Caroline; Schlapbach, Achim; Stachyra, Thérèse; Stutz, Stefan; Todorov, Milen; Jeay, Sébastien; Furet, Pascal Journal: Bioorganic & medicinal chemistry letters Issue: Volume 28:Issue 20(2018) Page Start: 3404 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
20. Molecular and structural characterization of a TEAD mutation at the origin of Sveinsson's chorioretinal atrophy. (11th April 2019) Authors: Bokhovchuk, Fedir; Mesrouze, Yannick; Izaac, Aude; Meyerhofer, Marco; Zimmermann, Catherine; Fontana, Patrizia; Schmelzle, Tobias; Erdmann, Dirk; Furet, Pascal; Kallen, Joerg; Chène, Patrick Journal: FEBS journal Issue: Volume 286:Number 12(2019) Page Start: 2381 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗