1. A poised fragment library enables rapid synthetic expansion yielding the first reported inhibitors of PHIP(2), an atypical bromodomain. Issue 3 (13th January 2016) Authors: Cox, Oakley B.; Krojer, Tobias; Collins, Patrick; Monteiro, Octovia; Talon, Romain; Bradley, Anthony; Fedorov, Oleg; Amin, Jahangir; Marsden, Brian D.; Spencer, John; von Delft, Frank; Brennan, Paul E. Journal: Chemical science Issue: Volume 7:Issue 3(2016:Mar.) Page Start: 2322 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced‐Fit Pocket Stabilized by a Cation–π Interaction1. (12th May 2014) Authors: Rooney, Timothy P. C.; Filippakopoulos, Panagis; Fedorov, Oleg; Picaud, Sarah; Cortopassi, Wilian A.; Hay, Duncan A.; Martin, Sarah; Tumber, Anthony; Rogers, Catherine M.; Philpott, Martin; Wang, Minghua; Thompson, Amber L.; Heightman, Tom D.; Pryde, David C.; Cook, Andrew; Paton, Robert S.; Müll... Journal: Angewandte Chemie Issue: Volume 126:Number 24(2014) Page Start: 6240 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced‐Fit Pocket Stabilized by a Cation–π Interaction1. Issue 24 (12th May 2014) Authors: Rooney, Timothy P. C.; Filippakopoulos, Panagis; Fedorov, Oleg; Picaud, Sarah; Cortopassi, Wilian A.; Hay, Duncan A.; Martin, Sarah; Tumber, Anthony; Rogers, Catherine M.; Philpott, Martin; Wang, Minghua; Thompson, Amber L.; Heightman, Tom D.; Pryde, David C.; Cook, Andrew; Paton, Robert S.; Müll... Journal: Angewandte Chemie international edition Issue: Volume 53:Issue 24(2014) Page Start: 6126 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. An Activity‐Based Probe Targeting Non‐Catalytic, Highly Conserved Amino Acid Residues within Bromodomains. (27th December 2018) Authors: D'Ascenzio, Melissa; Pugh, Kathryn M.; Konietzny, Rebecca; Berridge, Georgina; Tallant, Cynthia; Hashem, Shaima; Monteiro, Octovia; Thomas, Jason R.; Schirle, Markus; Knapp, Stefan; Marsden, Brian; Fedorov, Oleg; Bountra, Chas; Kessler, Benedikt M.; Brennan, Paul E. Journal: Angewandte Chemie Issue: Volume 131:Number 4(2019) Page Start: 1019 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. An Activity‐Based Probe Targeting Non‐Catalytic, Highly Conserved Amino Acid Residues within Bromodomains. Issue 4 (27th December 2018) Authors: D'Ascenzio, Melissa; Pugh, Kathryn M.; Konietzny, Rebecca; Berridge, Georgina; Tallant, Cynthia; Hashem, Shaima; Monteiro, Octovia; Thomas, Jason R.; Schirle, Markus; Knapp, Stefan; Marsden, Brian; Fedorov, Oleg; Bountra, Chas; Kessler, Benedikt M.; Brennan, Paul E. Journal: Angewandte Chemie international edition Issue: Volume 58:Issue 4(2019) Page Start: 1007 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Back Cover: Discovery of a PCAF Bromodomain Chemical Probe (Angew. Chem. Int. Ed. 3/2017). Issue 3 (23rd December 2016) Authors: Moustakim, Moses; Clark, Peter G. K.; Trulli, Laura; Fuentes de Arriba, Angel L.; Ehebauer, Matthias T.; Chaikuad, Apirat; Murphy, Emma J.; Mendez‐Johnson, Jacqui; Daniels, Danette; Hou, Chun‐Feng D.; Lin, Yu‐Hui; Walker, John R.; Hui, Raymond; Yang, Hongbing; Dorrell, Lucy; Rogers, Catherine M.;... Journal: Angewandte Chemie international edition Issue: Volume 56:Issue 3(2017) Page Start: 908 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. CBP/p300 Bromodomains Regulate Amyloid-like Protein Aggregation upon Aberrant Lysine Acetylation. Issue 1 (19th January 2017) Authors: Olzscha, Heidi; Fedorov, Oleg; Kessler, Benedikt M.; Knapp, Stefan; La Thangue, Nicholas B. Journal: Cell chemical biology Issue: Volume 24:Issue 1(2017) Page Start: 9 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Correction: Synthesis of kinase inhibitors containing a pentafluorosulfanyl moiety. Issue 2 (19th December 2017) Authors: Sansook, Supojjanee; Ocasio, Cory A.; Day, Iain J.; Tizzard, Graham J.; Coles, Simon J.; Fedorov, Oleg; Bennett, James M.; Elkins, Jonathan M.; Spencer, John Journal: Organic & biomolecular chemistry Issue: Volume 16:Issue 2(2017) Page Start: 336 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Design and synthesis of potent and selective inhibitors of BRD7 and BRD9 bromodomains1. Issue 7 (8th July 2015) Authors: Hay, Duncan A.; Rogers, Catherine M.; Fedorov, Oleg; Tallant, Cynthia; Martin, Sarah; Monteiro, Octovia P.; Müller, Susanne; Knapp, Stefan; Schofield, Christopher J.; Brennan, Paul E. Journal: MedChemComm Issue: Volume 6:Issue 7(2015:Jul.) Page Start: 1381 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. Design, Synthesis and Characterization of Covalent KDM5 Inhibitors. (7th December 2018) Authors: Vazquez‐Rodriguez, Saleta; Wright, Miranda; Rogers, Catherine M.; Cribbs, Adam P.; Velupillai, Srikannathasan; Philpott, Martin; Lee, Henry; Dunford, James E.; Huber, Kilian V. M.; Robers, Matthew B.; Vasta, James D.; Thezenas, Marie‐Laetitia; Bonham, Sarah; Kessler, Benedikt; Bennett, James; Fed... Journal: Angewandte Chemie Issue: Volume 131:Number 2(2019) Page Start: 525 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗