Search

Author/Creator Fan, Erkang

1. 5-Aminopyrazole-4-carboxamide analogues are selective inhibitors of Plasmodium falciparum microgametocyte exflagellation and potential malaria transmission blocking agents. Issue 22 (15th November 2016)

Authors:
Huang, Wenlin; Hulverson, Matthew A.; Zhang, Zhongsheng; Choi, Ryan; Hart, Kevin J.; Kennedy, Mark; Vidadala, Rama Subba Rao; Maly, Dustin J.; Van Voorhis, Wesley C.; Lindner, Scott E.; Fan, Erkang; Ojo, Kayode K.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 22(2016)
Page Start:
5487
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗

2. A binding hotspot in Trypanosoma cruzi histidyl‐tRNA synthetase revealed by fragment‐based crystallographic cocktail screens. (1st August 2015)

Authors:
Koh, Cho Yeow; Kallur Siddaramaiah, Latha; Ranade, Ranae M.; Nguyen, Jasmine; Jian, Tengyue; Zhang, Zhongsheng; Gillespie, J. Robert; Buckner, Frederick S.; Verlinde, Christophe L. M. J.; Fan, Erkang; Hol, Wim G. J.
Journal:
Acta crystallographica
Issue:
Volume 71:Part 8(2015:Aug.)
Page Start:
1684
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗

3. Bumped Kinase Inhibitors as therapy for apicomplexan parasitic diseases: lessons learned. Issue 5 (May 2020)

Authors:
Choi, Ryan; Hulverson, Matthew A.; Huang, Wenlin; Vidadala, Rama S.R.; Whitman, Grant R.; Barrett, Lynn K.; Schaefer, Deborah A.; Betzer, Dana P.; Riggs, Michael W.; Doggett, J. Stone; Hemphill, Andrew; Ortega-Mora, Luis Miguel; McCloskey, Molly C.; Arnold, Samuel L.M.; Hackman, Robert C.; Marsh,...
Journal:
International journal for parasitology
Issue:
Volume 50:Issue 5(2020)
Page Start:
413
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗

8. Identification of Potent Inhibitors of the Trypanosoma brucei Methionyl-tRNA Synthetase via High-Throughput Orthogonal Screening. (January 2015)

Authors:
Pedró-Rosa, Laura; Buckner, Frederick S.; Ranade, Ranae M.; Eberhart, Christina; Madoux, Franck; Gillespie, J. Robert; Koh, Cho Yeow; Brown, Steven; Lohse, Jacqueline; Verlinde, Christophe L. M.; Fan, Erkang; Bannister, Thomas; Scampavia, Louis; Hol, Wim G. J.; Spicer, Timothy; Hodder, Peter
Journal:
Journal of biomolecular screening
Issue:
Volume 20:Number 1(2015)
Page Start:
122
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗

9. In vitro efficacy of bumped kinase inhibitors against Besnoitia besnoiti tachyzoites. Issue 12 (October 2017)

Authors:
Jiménez-Meléndez, Alejandro; Ojo, Kayode K.; Wallace, Alexandra M.; Smith, Tess R.; Hemphill, Andrew; Balmer, Vreni; Regidor-Cerrillo, Javier; Ortega-Mora, Luis M.; Hehl, Adrian B.; Fan, Erkang; Maly, Dustin J.; Van Voorhis, Wesley C.; Álvarez-García, Gema
Journal:
International journal for parasitology
Issue:
Volume 47:Issue 12(2017)
Page Start:
811
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗

10. Methionyl-tRNA synthetase inhibitor has potent in vivo activity in a novel Giardia lamblia luciferase murine infection model. (3rd February 2020)

Authors:
Michaels, Samantha A; Shih, Han-Wei; Zhang, Bailin; Navaluna, Edelmar D; Zhang, Zhongsheng; Ranade, Ranae M; Gillespie, J Robert; Merritt, Ethan A; Fan, Erkang; Buckner, Frederick S; Paredez, Alexander R; Ojo, Kayode K
Journal:
Journal of antimicrobial chemotherapy
Issue:
Volume 75:Number 5(2020)
Page Start:
1218
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗