1. 3-Substituted Quinolines as RORγt Inverse Agonists. Issue 12 (15th June 2019) Authors: Tanis, Virginia M.; Venkatesan, Hariharan; Cummings, Maxwell D.; Albers, Michael; Kent Barbay, J.; Herman, Krystal; Kummer, David A.; Milligan, Cynthia; Nelen, Marina I.; Nishimura, Rachel; Schlueter, Thomas; Scott, Brian; Spurlino, John; Wolin, Ronald; Woods, Craig; Xue, Xiaohua; Edwards, James ... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 29:Issue 12(2019) Page Start: 1463 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. 6-Substituted quinolines as RORγt inverse agonists. Issue 23 (1st December 2017) Authors: Barbay, J. Kent; Cummings, Maxwell D.; Abad, Marta; Castro, Glenda; Kreutter, Kevin D.; Kummer, David A.; Maharoof, Umar; Milligan, Cynthia; Nishimura, Rachel; Pierce, Joan; Schalk-Hihi, Celine; Spurlino, John; Tanis, Virginia M.; Urbanski, Maud; Venkatesan, Hariharan; Wang, Aihua; Woods, Craig; ... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 23(2017) Page Start: 5277 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. A carboxylic acid isostere screen of the DHODH inhibitor Brequinar. Issue 22 (15th November 2020) Authors: DeRatt, Lindsey G.; Christine Pietsch, E.; Tanner, Alexandra; Shaffer, Paul; Jacoby, Edgar; Wang, Weixue; Kazmi, Faraz; Zhang, Xiaochun; Attar, Ricardo M.; Edwards, James P.; Kuduk, Scott D. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 30:Issue 22(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Assessing IRAK4 Functions in ABC DLBCL by IRAK4 Kinase Inhibition and Protein Degradation. Issue 12 (17th December 2020) Authors: Zhang, Jing; Fu, Liqiang; Shen, Bin; Liu, Yingtao; Wang, Wenqian; Cai, Xin; Kong, Linglong; Yan, Yilin; Meng, Ryan; Zhang, Zhuming; Chen, Ying-Nan P.; Liu, Qian; Wan, Zhao-Kui; Zhou, Tianyuan; Wang, Xiaotao; Gavine, Paul; Del Rosario, Amanda; Ahn, Kay; Philippar, Ulrike; Attar, Ricardo Journal: Cell chemical biology Issue: Volume 27:Issue 12(2020) Page Start: 1500 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Diaminopyrimidines, diaminopyridines and diaminopyridazines as histamine H4 receptor modulators. Issue 4 (15th February 2015) Authors: Savall, Brad M.; Meduna, Steven P.; Tays, Kevin; Cai, Hui; Thurmond, Robin L.; McGovern, Patricia; Gaul, Michael; Zhao, Bao-Ping; Edwards, James P. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 4(2015) Page Start: 956 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Discovery and optimization of new oxadiazole substituted thiazole RORγt inverse agonists through a bioisosteric amide replacement approach. Issue 12 (15th June 2020) Authors: Steeneck, Christoph; Gege, Christian; Kinzel, Olaf; Albers, Michael; Kleymann, Gerald; Schlüter, Thomas; Schulz, Andreas; Xue, Xiaohua; Cummings, Maxwell D.; Fourie, Anne M.; Leonard, Kristi A.; Scott, Brian; Edwards, James P.; Hoffmann, Thomas; Goldberg, Steven D. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 30:Issue 12(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Identification and biological evaluation of thiazole-based inverse agonists of RORγt. Issue 9 (15th May 2018) Authors: Gege, Christian; Cummings, Maxwell D.; Albers, Michael; Kinzel, Olaf; Kleymann, Gerald; Schlüter, Thomas; Steeneck, Christoph; Nelen, Marina I.; Milligan, Cindy; Spurlino, John; Xue, Xiaohua; Leonard, Kristi; Edwards, James P.; Fourie, Anne; Goldberg, Steven D.; Hoffmann, Thomas Journal: Bioorganic & medicinal chemistry letters Issue: Volume 28:Issue 9(2018) Page Start: 1446 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Identification and structure activity relationships of quinoline tertiary alcohol modulators of RORγt. Issue 9 (1st May 2017) Authors: Kummer, David A.; Cummings, Maxwell D.; Abad, Marta; Barbay, Joseph; Castro, Glenda; Wolin, Ronald; Kreutter, Kevin D.; Maharoof, Umar; Milligan, Cynthia; Nishimura, Rachel; Pierce, Joan; Schalk-Hihi, Celine; Spurlino, John; Urbanski, Maud; Venkatesan, Hariharan; Wang, Aihua; Woods, Craig; Xue, X... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 9(2017) Page Start: 2047 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Immunological characterization of HM5023507, an orally active PI3Kδ/γ inhibitor. Issue 1 (13th January 2020) Authors: Cai, Yu; Yu, Jun; Ren, Ping; He, Jianlin; Wu, Zhipeng; Xiao, Kun; Jia, Hong; Wang, Jian; Sai, Yang; Dai, Guangxiu; Li, Xiong; Su, Weiguo; Ngo, Karen; Castro, Glenda; Acton, Paul D.; Fung‐Leung, Wai‐Ping; Edwards, James P.; Venable, Jennifer; Rao, Tadimeti S. Journal: Pharmacology research & perspectives Issue: Volume 8:Issue 1(2020) Page Start: n/a Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. Optimization and biological evaluation of thiazole-bis-amide inverse agonists of RORγt. Issue 12 (15th June 2020) Authors: Gege, Christian; Albers, Michael; Kinzel, Olaf; Kleymann, Gerald; Schlüter, Thomas; Steeneck, Christoph; Hoffmann, Thomas; Xue, Xiaohua; Cummings, Maxwell D.; Spurlino, John; Milligan, Cynthia; Fourie, Anne M.; Edwards, James P.; Leonard, Kristi; Coe, Kevin; Scott, Brian; Pippel, Dan; Goldberg, S... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 30:Issue 12(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗