1. Azepino-indazoles as calcitonin gene-related peptide (CGRP) receptor antagonists. (1st January 2021) Authors: Mercer, Stephen E.; Chaturvedula, Prasad V.; Conway, Charles M.; Cook, Deborah A.; Davis, Carl D.; Pin, Sokhom S.; Macci, Robert; Schartman, Richard; Signor, Laura J.; Widmann, Kimberly A.; Whiterock, Valerie J.; Chen, Ping; Xu, Cen; Herbst, John J.; Kostich, Walter A.; Thalody, George; Macor, Jo... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 31(2021) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Calcitonin gene-related peptide (CGRP) receptor antagonists: Heterocyclic modification of a novel azepinone lead. (1st July 2021) Authors: Luo, Guanglin; Jiang, Xiang-Jun; Chen, Ling; Conway, Charles M.; Gulianello, Michael; Kostich, Walter; Keavy, Deborah; Signor, Laura J.; Chen, Ping; Davis, Carl; Whiterock, Valerie J.; Schartman, Richard; Widmann, Kimberly A.; Macor, John E.; Dubowchik, Gene M. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 43(2021) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Discovery of new acylaminopyridines as GSK-3 inhibitors by a structure guided in-depth exploration of chemical space around a pyrrolopyridinone core. Issue 9 (1st May 2015) Authors: Sivaprakasam, Prasanna; Han, Xiaojun; Civiello, Rita L.; Jacutin-Porte, Swanee; Kish, Kevin; Pokross, Matt; Lewis, Hal A.; Ahmed, Nazia; Szapiel, Nicolas; Newitt, John A.; Baldwin, Eric T.; Xiao, Hong; Krause, Carol M.; Park, Hyunsoo; Nophsker, Michelle; Lippy, Jonathan S.; Burton, Catherine R.; ... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 9(2015) Page Start: 1856 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Discovery of new acylaminopyridines as GSK-3 inhibitors by a structure guided in-depth exploration of chemical space around a pyrrolopyridinone core. Issue 9 (1st May 2015) Authors: Sivaprakasam, Prasanna; Han, Xiaojun; Civiello, Rita L.; Jacutin-Porte, Swanee; Kish, Kevin; Pokross, Matt; Lewis, Hal A.; Ahmed, Nazia; Szapiel, Nicolas; Newitt, John A.; Baldwin, Eric T.; Xiao, Hong; Krause, Carol M.; Park, Hyunsoo; Nophsker, Michelle; Lippy, Jonathan S.; Burton, Catherine R.; ... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 9(2015) Page Start: 1856 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Structure–activity relationship (SAR) studies on substituted N-(pyridin-3-yl)-2-amino-isonicotinamides as highly potent and selective glycogen synthase kinase-3 (GSK-3) inhibitors. (1st February 2023) Authors: Luo, Guanglin; Chen, Ling; Jacutin-Porte, Swanee; Han, Ying; Burton, Catherine R.; Xiao, Hong; Krause, Carol M.; Cao, Yang; Liu, Nengyin; Kish, Kevin; Lewis, Hal A.; Macor, John E.; Dubowchik, Gene M. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 81(2023) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Synthesis and SAR of calcitonin gene-related peptide (CGRP) antagonists containing substituted aryl-piperazines and piperidines. Issue 4 (15th February 2016) Authors: Civiello, Rita L.; Han, Xiaojun; Beno, Brett R.; Chaturvedula, Prasad V.; Herbst, John J.; Xu, Cen; Conway, Charles M.; Macor, John E.; Dubowchik, Gene M. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 4(2016) Page Start: 1229 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗