Discovery of new acylaminopyridines as GSK-3 inhibitors by a structure guided in-depth exploration of chemical space around a pyrrolopyridinone core. Issue 9 (1st May 2015)

• Record Type: Journal Article
• Authors: Sivaprakasam, Prasanna; Han, Xiaojun; Civiello, Rita L.; Jacutin-Porte, Swanee; Kish, Kevin; Pokross, Matt; Lewis, Hal A.; Ahmed, Nazia; Szapiel, Nicolas; Newitt, John A.; Baldwin, Eric T.; Xiao, Hong; Krause, Carol M.; Park, Hyunsoo; Nophsker, Michelle; Lippy, Jonathan S.; Burton, Catherine R.; Langley, David R.; Macor, John E.; Dubowchik, Gene M.
• Is Part Of: Bioorganic & medicinal chemistry letters. Volume 25:Issue 9(2015)
• Page Start: 1856
• Page End: 1863
• Publication Date: 2015-05-01
• Subjects: Bioorganic chemistry -- Periodicals; Pharmaceutical chemistry -- Periodicals; 572
• DOI: 10.1016/j.bmcl.2015.03.046
• Languages: English
• ISSNs: 0960-894X

Abstract

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