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Author/Creator Demarest, Keith

2. Canagliflozin: a sodium glucose co‐transporter 2 inhibitor for the treatment of type 2 diabetes mellitus. Issue 1 (25th August 2015)

Authors:
Rosenthal, Norm; Meininger, Gary; Ways, Kirk; Polidori, David; Desai, Mehul; Qiu, Rong; Alba, Maria; Vercruysse, Frank; Balis, Dainius; Shaw, Wayne; Edwards, Robert; Bull, Scott; Di Prospero, Nicholas; Sha, Sue; Rothenberg, Paul; Canovatchel, William; Demarest, Keith
Journal:
Annals of the New York Academy of Sciences
Issue:
Volume 1358:Issue 1(2015)
Page Start:
28
Record Type:
Journal Article
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3. Design, synthesis and biological evaluation of (2S, 3R, 4R, 5S, 6R)-5-fluoro-6-(hydroxymethyl)-2-aryltetrahydro-2H-pyran-3, 4-diols as potent and orally active SGLT dual inhibitors. Issue 21 (15th November 2018)

Authors:
Xu, Guozhang; Gaul, Michael D.; Kuo, Gee-Hong; Du, Fuyong; Xu, June Zhi; Wallace, Nathaniel; Hinke, Simon; Kirchner, Thomas; Silva, Jose; Huebert, Norman D.; Lee, Seunghun; Murray, William; Liang, Yin; Demarest, Keith
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 28:Issue 21(2018)
Page Start:
3446
Record Type:
Journal Article
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4. Design, synthesis and structure activity relationships of indazole and indole derivatives as potent glucagon receptor antagonists. Issue 15 (1st August 2019)

Authors:
Song, Fengbin; Xu, Guozhang; Gaul, Michael D.; Zhao, Baoping; Lu, Tianbao; Zhang, Rui; DesJarlais, Renee L.; DiLoreto, Karen; Huebert, Norman; Shook, Brian; Rentzeperis, Dennis; Santulli, Rosie; Eckardt, Annette; Demarest, Keith
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 29:Issue 15(2019)
Page Start:
1974
Record Type:
Journal Article
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5. Discovery of potent and orally bioavailable indazole-based glucagon receptor antagonists for the treatment of type 2 diabetes. Issue 20 (15th October 2019)

Authors:
Xu, Guozhang; Gaul, Michael D.; Song, Fengbin; Du, Fuyong; Liang, Yin; DesJarlais, Renee L.; DiLoreto, Karen; Shook, Brian; Rentzeperis, Dennis; Santulli, Rosie; Eckardt, Annette; Demarest, Keith
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 29:Issue 20(2019)
Page Start:
Record Type:
Journal Article
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6. Evaluation of anti-diabetic effect and gall bladder function with 2-thio-5-thiomethyl substituted imidazoles as TGR5 receptor agonists. Issue 8 (15th April 2017)

Authors:
Zhang, Xuqing; Sui, Zhihua; Kauffman, Jack; Hou, Cuifen; Chen, Cailin; Du, Fuyong; Kirchner, Thomas; Liang, Yin; Johnson, Dana; Murray, William V.; Demarest, Keith
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 8(2017)
Page Start:
1760
Record Type:
Journal Article
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7. Synthesis and biological evaluation of benzocyclobutane-C-glycosides as potent and orally active SGLT1/SGLT2 dual inhibitors. Issue 7 (15th April 2018)

Authors:
Kuo, Gee-Hong; Gaul, Micheal D.; Liang, Yin; Xu, June Z.; Du, Fuyong; Hornby, Pamela; Xu, Guozhang; Qi, Jenson; Wallace, Nathaniel; Lee, Seunghun; Grant, Eugene; Murray, William V.; Demarest, Keith
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 28:Issue 7(2018)
Page Start:
1182
Record Type:
Journal Article
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