1. Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation. (1st January 2020) Authors: Fois, Benedetta; Distinto, Simona; Meleddu, Rita; Deplano, Serenella; Maccioni, Elias; Floris, Costantino; Rosa, Antonella; Nieddu, Mariella; Caboni, Pierluigi; Sissi, Claudia; Angeli, Andrea; Supuran, Claudiu T.; Cottiglia, Filippo Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 35:Number 1(2020) Page Start: 539 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Design, Synthesis, and Biological Evaluation of 1, 3‐Diarylpropenones as Dual Inhibitors of HIV‐1 Reverse Transcriptase. Issue 8 (21st May 2014) Authors: Meleddu, Rita; Cannas, Valeria; Distinto, Simona; Sarais, Giorgia; Del Vecchio, Claudia; Esposito, Francesca; Bianco, Giulia; Corona, Angela; Cottiglia, Filippo; Alcaro, Stefano; Parolin, Cristina; Artese, Anna; Scalise, Daniela; Fresta, Massimo; Arridu, Antonella; Ortuso, Francesco; Maccioni, El... Journal: ChemMedChem Issue: Volume 9:Issue 8(2014:Aug.) Page Start: 1869 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Exploring new structural features of the 4-[(3-methyl-4-aryl-2, 3-dihydro-1, 3-thiazol-2-ylidene)amino]benzenesulphonamide scaffold for the inhibition of human carbonic anhydrases. (1st January 2019) Authors: Distinto, Simona; Meleddu, Rita; Ortuso, Francesco; Cottiglia, Filippo; Deplano, Serenella; Sequeira, Lisa; Melis, Claudia; Fois, Benedetta; Angeli, Andrea; Capasso, Clemente; Angius, Rossella; Alcaro, Stefano; Supuran, Claudiu T.; Maccioni, Elias Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 34:Number 1(2019) Page Start: 1526 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Exploring the thiazole scaffold for the identification of new agents for the treatment of fluconazole resistant Candida. (1st November 2016) Authors: Meleddu, Rita; Distinto, Simona; Corona, Angela; Maccioni, Elias; Arridu, Antonella; Melis, Claudia; Bianco, Giulia; Matyus, Peter; Cottiglia, Filippo; Sanna, Adriana; De Logu, Alessandro Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 31:Number 6(2016:Dec.) Page Start: 1672 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Flavonoids and Acid-Hydrolysis derivatives of Neo-Clerodane diterpenes from Teucrium flavum subsp. glaucum as inhibitors of the HIV-1 reverse transcriptase–associated RNase H function. (1st January 2021) Authors: Fois, Benedetta; Corona, Angela; Tramontano, Enzo; Distinto, Simona; Maccioni, Elias; Meleddu, Rita; Caboni, Pierluigi; Floris, Costantino; Cottiglia, Filippo Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 36:Number 1(2021) Page Start: 749 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Isatin thiazoline hybrids as dual inhibitors of HIV-1 reverse transcriptase. (1st January 2017) Authors: Meleddu, Rita; Distinto, Simona; Corona, Angela; Tramontano, Enzo; Bianco, Giulia; Melis, Claudia; Cottiglia, Filippo; Maccioni, Elias Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 32:Number 1(2017) Page Start: 130 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Isatin: a privileged scaffold for the design of carbonic anhydrase inhibitors. (1st January 2017) Authors: Melis, Claudia; Meleddu, Rita; Angeli, Andrea; Distinto, Simona; Bianco, Giulia; Capasso, Clemente; Cottiglia, Filippo; Angius, Rossella; Supuran, Claudiu T.; Maccioni, Elias Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 32:Number 1(2017) Page Start: 68 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. New 4-[(3-cyclohexyl-4-aryl-2, 3-dihydro-1, 3-thiazol-2-ylidene)amino]benzene-1-sulfonamides, synthesis and inhibitory activity toward carbonic anhydrase I, II, IX, XII. Issue 16 (15th August 2015) Authors: Meleddu, Rita; Maccioni, Elias; Distinto, Simona; Bianco, Giulia; Melis, Claudia; Alcaro, Stefano; Cottiglia, Filippo; Ceruso, Mariangela; Supuran, Claudiu T. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 16(2015) Page Start: 3281 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. New 4-[(3-cyclohexyl-4-aryl-2, 3-dihydro-1, 3-thiazol-2-ylidene)amino]benzene-1-sulfonamides, synthesis and inhibitory activity toward carbonic anhydrase I, II, IX, XII. Issue 16 (15th August 2015) Authors: Meleddu, Rita; Maccioni, Elias; Distinto, Simona; Bianco, Giulia; Melis, Claudia; Alcaro, Stefano; Cottiglia, Filippo; Ceruso, Mariangela; Supuran, Claudiu T. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 16(2015) Page Start: 3281 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. Selective inhibition of carbonic anhydrase IX and XII by coumarin and psoralen derivatives. (1st January 2021) Authors: Meleddu, Rita; Deplano, Serenella; Maccioni, Elias; Ortuso, Francesco; Cottiglia, Filippo; Secci, Daniela; Onali, Alessia; Sanna, Erica; Angeli, Andrea; Angius, Rossella; Alcaro, Stefano; Supuran, Claudiu T.; Distinto, Simona Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 36:Number 1(2021) Page Start: 685 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗