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Author/Creator Chase, Peter

1. Discovery and SAR of a novel series of potent, CNS penetrant M4 PAMs based on a non-enolizable ketone core: Challenges in disposition. Issue 17 (1st September 2016)

Authors:
Wood, Michael R.; Noetzel, Meredith J.; Tarr, James C.; Rodriguez, Alice L.; Lamsal, Atin; Chang, Sichen; Foster, Jarrett J.; Smith, Emery; Chase, Peter; Hodder, Peter S.; Engers, Darren W.; Niswender, Colleen M.; Brandon, Nicholas J.; Wood, Michael W.; Duggan, Mark E.; Conn, P. Jeffrey; Bridges,...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 17(2016)
Page Start:
4282
Record Type:
Journal Article
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Available online (eLD content is only available in our Reading Rooms) ↗

5. Development of an HTS-Compatible Assay for Discovery of Melanoma-Related Microphthalmia Transcription Factor Disruptors Using AlphaScreen Technology. (January 2017)

Authors:
Wang, Jing; Fang, Pengfei; Chase, Peter; Tshori, Sagi; Razin, Ehud; Spicer, Timothy P.; Scampavia, Louis; Hodder, Peter; Guo, Min
Journal:
Journal of biomolecular screening
Issue:
Volume 22:Number 1(2017)
Page Start:
58
Record Type:
Journal Article
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6. An Ultra-High-Throughput Screen for Catalytic Inhibitors of Serine/Threonine Protein Phosphatases Types 1 and 5 (PP1C and PP5C). (January 2017)

Authors:
Swingle, Mark; Volmar, Claude-Henry; Saldanha, S. Adrian; Chase, Peter; Eberhart, Christina; Salter, Edward A.; D'Arcy, Brandon; Schroeder, Chad E.; Golden, Jennifer E.; Wierzbicki, Andrzej; Hodder, Peter; Honkanen, Richard E.
Journal:
Journal of biomolecular screening
Issue:
Volume 22:Number 1(2017)
Page Start:
21
Record Type:
Journal Article
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7. Discovery and optimization of a novel series of highly CNS penetrant M4 PAMs based on a 5, 6-dimethyl-4-(piperidin-1-yl)thieno[2, 3-d]pyrimidine core. Issue 13 (1st July 2016)

Authors:
Wood, Michael R.; Noetzel, Meredith J.; Engers, Julie L.; Bollinger, Katrina A.; Melancon, Bruce J.; Tarr, James C.; Han, Changho; West, Mary; Gregro, Alison R.; Lamsal, Atin; Chang, Sichen; Ajmera, Sonia; Smith, Emery; Chase, Peter; Hodder, Peter S.; Bubser, Michael; Jones, Carrie K.; Hopkins, C...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 13(2016)
Page Start:
3029
Record Type:
Journal Article
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8. Discovery and SAR of muscarinic receptor subtype 1 (M1) allosteric activators from a molecular libraries high throughput screen. Part 1: 2, 5-Dibenzyl-2H-pyrazolo[4, 3-c]quinolin-3(5H)-ones as positive allosteric modulators. Issue 2 (15th January 2015)

Authors:
Han, Changho; Chatterjee, Arindam; Noetzel, Meredith J.; Panarese, Joseph D.; Smith, Emery; Chase, Peter; Hodder, Peter; Niswender, Colleen; Conn, P. Jeffrey; Lindsley, Craig W.; Stauffer, Shaun R.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 25:Issue 2(2015)
Page Start:
384
Record Type:
Journal Article
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10. Fluorometric High-Throughput Screening Assay for Secreted Phospholipases A2 Using Phospholipid Vesicles. (August 2016)

Authors:
Ewing, Heather; Fernández-Vega, Virneliz; Spicer, Timothy P.; Chase, Peter; Brown, Steven; Scampavia, Louis; Roush, William R.; Riley, Sean; Rosen, Hugh; Hodder, Peter; Lambeau, Gerard; Gelb, Michael H.
Journal:
Journal of biomolecular screening
Issue:
Volume 21:Number 7(2016)
Page Start:
713
Record Type:
Journal Article
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