1. A convenient one-pot synthesis of boroxoles from diboronic acid. Issue 39 (27th September 2017) Authors: Lafitte, Guillaume; Kunihiro, Kana; Bonneaud, Céline; Dréan, Bénédicte; Gaigne, Frédéric; Parnet, Véronique; Pierre, Romain; Raffin, Catherine; Vatinel, Rodolphe; Fournier, Jean-François; Musicki, Branislav; Ouvry, Gilles; Bouix-Peter, Claire; Tomas, Loic; Harris, Craig S. Journal: Tetrahedron letters Issue: Volume 58:Issue 39(2017) Page Start: 3757 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. A facile and rapid preparation of hydroxamic acids by hydroxylaminolysis using DBU as base. Issue 20 (18th May 2016) Authors: Beillard, Audrey; Bhurruth-Alcor, Yushma; Bouix-Peter, Claire; Bouquet, Karinne; Chambon, Sandrine; Clary, Laurence; Harris, Craig S.; Millois, Corinne; Mouis, Grégoire; Ouvry, Gilles; Pierre, Romain; Reitz, Arnaud; Tomas, Loic Journal: Tetrahedron letters Issue: Volume 57:Issue 20(2016) Page Start: 2165 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. An efficient multi-component synthesis of N-1-alkylated 5-nitrouracils from α-amino acids. Issue 22 (1st June 2016) Authors: Boiteau, Jean-Guy; Bouix-Peter, Claire; Chambon, Sandrine; Clary, Laurence; Daver, Sebastien; Dumais, Laurence; Fournier, Jean-François; Harris, Craig S.; Mebrouk, Kenny; Millois, Corinne; Pierre, Romain; Rodeville, Nicolas; Talano, Sandrine; Tomas, Loïc Journal: Tetrahedron letters Issue: Volume 57:Issue 22(2016) Page Start: 2367 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. An expedient synthesis of non-racemic N-alkylated pyrrolidin-2, 5-diones and piperidin-2, 6-diones as peptidomimetics. Issue 52 (28th December 2016) Authors: Brethon, Anne; Bouix-Peter, Claire; Clary, Laurence; Fournier, Jean-François; Harris, Craig S.; Lardy, Claude; Roche, Didier; Rodeschini, Vincent; Talano, Sandrine Journal: Tetrahedron letters Issue: Volume 57:Issue 52(2016) Page Start: 5924 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Discovery and process development of a novel TACE inhibitor for the topical treatment of psoriasis. Issue 4 (15th February 2018) Authors: Boiteau, Jean-Guy; Ouvry, Gilles; Arlabosse, Jean-Marie; Astri, Stéphanie; Beillard, Audrey; Bhurruth-Alcor, Yushma; Bonnary, Laetitia; Bouix-Peter, Claire; Bouquet, Karine; Bourotte, Marilyne; Cardinaud, Isabelle; Comino, Catherine; Deprez, Benoît; Duvert, Denis; Féret, Angélique; Hacini-Rachine... Journal: Bioorganic & medicinal chemistry Issue: Volume 26:Issue 4(2018) Page Start: 945 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Discovery of phenoxyindazoles and phenylthioindazoles as RORγ inverse agonists. Issue 23 (1st December 2016) Authors: Ouvry, Gilles; Bouix-Peter, Claire; Ciesielski, Fabrice; Chantalat, Laurent; Christin, Olivier; Comino, Catherine; Duvert, Denis; Feret, Christophe; Harris, Craig S.; Lamy, Laurent; Luzy, Anne-Pascale; Musicki, Branislav; Orfila, Danielle; Pascau, Jonathan; Parnet, Véronique; Perrin, Agnès; Pierr... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 23(2016) Page Start: 5802 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Identification of novel TACE inhibitors compatible with topical application. Issue 8 (15th April 2017) Authors: Ouvry, Gilles; Berton, Yaël; Bhurruth-Alcor, Yushma; Bonnary, Laetitia; Bouix-Peter, Claire; Bouquet, Karine; Bourotte, Marilyne; Chambon, Sandrine; Comino, Catherine; Deprez, Benoît; Duvert, Denis; Duvert, Gwenaëlle; Hacini-Rachinel, Feriel; Harris, Craig S.; Luzy, Anne-Pascale; Mathieu, Arnaud;... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 8(2017) Page Start: 1848 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. N-3 alkylation of uracils with unprotected amino alcohols using the Mitsunobu reaction. Issue 3 (17th January 2018) Authors: Lafitte, Guillaume; Beillard, Audrey; Chambon, Sandrine; Soulet, Catherine; Dumais, Laurence; Mouis, Grégoire; Fournier, Jean-François; Clary, Laurence; Bouix-Peter, Claire; Tomas, Loic; Harris, Craig S. Journal: Tetrahedron letters Issue: Volume 59:Issue 3(2018) Page Start: 256 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Route scouting and optimization of a potent sulfoximine-based inverse agonist of RORγt. Issue 40 (4th October 2018) Authors: Lafitte, Guillaume; Parnet, Veronique; Pierre, Romain; Raffin, Catherine; Vatinel, Rodolphe; Musicki, Branislav; Tomas, Loic; Bouix-Peter, Claire; Ouvry, Gilles; Daver, Sebastien; Arlabosse, Jean-Marie; Boiteau, Jean-Guy; Gerfaud, Thibaud; Harris, Craig S. Journal: Tetrahedron Issue: Volume 74:Issue 40(2018) Page Start: 5974 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. Squaramides as novel class I and IIB histone deacetylase inhibitors for topical treatment of cutaneous t-cell lymphoma. Issue 17 (15th September 2018) Authors: Fournier, Jean-François; Bhurruth-Alcor, Yushma; Musicki, Branislav; Aubert, Jérome; Aurelly, Michèle; Bouix-Peter, Claire; Bouquet, Karinne; Chantalat, Laurent; Delorme, Marion; Drean, Bénédicte; Duvert, Gwenaelle; Fleury-Bregeot, Nicolas; Gauthier, Blanche; Grisendi, Karine; Harris, Craig S.; H... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 28:Issue 17(2018) Page Start: 2985 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗