Ligand-controlled regiodivergent direct arylation of indoles via oxidative boron Heck reaction. Issue 21 (21st September 2022) - Yang, Yo-Sep
Abstract : Ligand-controlled direct arylation of indoles via Pd(ii ) catalyzed oxidative boron Heck reaction under aerobic conditions is reported. Abstract : Ligand-controlled direct arylation of indoles via Pd(ii ) catalyzed oxidative boron Heck reaction under aerobic conditions is reported. This methodology provides a regiodivergent route for C2 or C3 aryl indoles in a protection free and acid/base free manner.