DBU-catalyzed Michael addition of bulky glycine imine to α, β-unsaturated isoxazoles and pyrazolamides. (19th November 2021)
- Record Type:
- Journal Article
- Title:
- DBU-catalyzed Michael addition of bulky glycine imine to α, β-unsaturated isoxazoles and pyrazolamides. (19th November 2021)
- Main Title:
- DBU-catalyzed Michael addition of bulky glycine imine to α, β-unsaturated isoxazoles and pyrazolamides
- Authors:
- Bai, Yu-Jun
Hu, Xiao-Mu
Bai, Ya-Jun
Zheng, Xiao-Hui
Zhang, Sheng-Yong
Ping-AnWang, - Abstract:
- Graphical abstract: DBU-catalyzed Michael additions of bulky glycine imines to α, β-unsaturated isoxazoles and pyrazolamides have been realized in THF with 1.0 eq. LiBr as an additive at room temperature to provide Michael adducts in excellent yields (up to 97%) and diastereoselectivities (> 20:1). Image 1
- Is Part Of:
- Tetrahedron. Volume 101(2021)
- Journal:
- Tetrahedron
- Issue:
- Volume 101(2021)
- Issue Display:
- Volume 101, Issue 2021 (2021)
- Year:
- 2021
- Volume:
- 101
- Issue:
- 2021
- Issue Sort Value:
- 2021-0101-2021-0000
- Page Start:
- Page End:
- Publication Date:
- 2021-11-19
- Subjects:
- Michael addition -- Glycine imine -- α, β-unsaturated isoxazole -- α, β-unsaturated pyrazolamide -- 1, 8-Diazabicyclo[5.4.0]undec-7-ene (DBU)
Chemistry, Organic -- Periodicals
547.005 - Journal URLs:
- http://www.elsevier.com/journals ↗
- DOI:
- 10.1016/j.tet.2021.132511 ↗
- Languages:
- English
- ISSNs:
- 0040-4020
- Deposit Type:
- Legaldeposit
- View Content:
- Available online (eLD content is only available in our Reading Rooms) ↗
- Physical Locations:
- British Library DSC - 8796.850000
British Library DSC - BLDSS-3PM
British Library STI - ELD Digital store - Ingest File:
- 19786.xml