ChemInform Abstract: Chiral Phosphoric Acid Catalyzed Highly Enantioselective Friedel—Crafts Alkylation Reaction of C3‐Substituted Indoles to β, γ‐Unsaturated α‐Ketimino Esters. Issue 25 (5th June 2015)

• Record Type: Journal Article
• Authors: Bi, Bo; Lou, Qin‐Xin; Ding, Yu‐Yang; Chen, Sheng‐Wei; Zhang, Sha‐Sha; Hu, Wen‐Hui; Zhao, Jun‐Ling
• Is Part Of: ChemInform. Volume 46:Issue 25(2015)
• Page Start: no
• Page End: no
• Publication Date: 2015-06-05
• Subjects: oxazine derivatives -- indole derivatives, isoindole derivatives -- diastereoselective syntheses, enantioselective syntheses (incl. cis/trans‐isomerism) -- catalysis, phase‐transfer catalysis; Chemistry -- Abstracts -- Periodicals; 540.5
• DOI: 10.1002/chin.201525213
• Languages: English
• ISSNs: 0931-7597

Abstract

Abstract: The scalable reaction allows the preparation of C2‐substituted indole derivatives bearing an α‐ketimino ester motif in moderate to high yields.