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    Igawa, H. et al. (2016). Amine-free melanin-concentrating hormone receptor 1 antagonists: Novel 1-(1H-benzimidazol-6-yl)pyridin-2(1H)-one derivatives and design to avoid CYP3A4 time-dependent inhibition. Bioorganic & medicinal chemistry. 24 (11), pp. 2486-2503. [Online]. 
  
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