1, 3-Iodo-amination of 2-methyl indoles via Csp2–Csp3 dual functionalization with iodine reagent. Issue 34 (19th February 2018)
- Record Type:
- Journal Article
- Title:
- 1, 3-Iodo-amination of 2-methyl indoles via Csp2–Csp3 dual functionalization with iodine reagent. Issue 34 (19th February 2018)
- Main Title:
- 1, 3-Iodo-amination of 2-methyl indoles via Csp2–Csp3 dual functionalization with iodine reagent
- Authors:
- Moriyama, Katsuhiko
Hamada, Tsukasa
Ishida, Kazuma
Togo, Hideo - Abstract:
- Abstract : Remote iodo-amination of indole derivatives via Csp 2 –Csp 3 dual functionalization under transition-metal-free conditions. Abstract : A 1, 3-iodo-amination with iodine reagent that involved the Csp 2 –Csp 3 dual functionalization of 2-methyl indoles was developed to provide 2-aminomethyl-3-iodo-indole derivatives. The iodo-amination proceeded via a 1, 4-transfer of an imide group through the formation of an indolyl(phenyl)iodonium imide using PhI(OAc)2, followed by an iodination using DIH or a double iodination of indole using excess DIH.
- Is Part Of:
- Chemical communications. Volume 54:Issue 34(2018)
- Journal:
- Chemical communications
- Issue:
- Volume 54:Issue 34(2018)
- Issue Display:
- Volume 54, Issue 34 (2018)
- Year:
- 2018
- Volume:
- 54
- Issue:
- 34
- Issue Sort Value:
- 2018-0054-0034-0000
- Page Start:
- 4258
- Page End:
- 4261
- Publication Date:
- 2018-02-19
- Subjects:
- Chemistry -- Periodicals
540 - Journal URLs:
- http://pubs.rsc.org/en/journals/journalissues/cc ↗
http://www.rsc.org/ ↗ - DOI:
- 10.1039/c8cc00352a ↗
- Languages:
- English
- ISSNs:
- 1359-7345
- Deposit Type:
- Legaldeposit
- View Content:
- Available online (eLD content is only available in our Reading Rooms) ↗
- Physical Locations:
- British Library DSC - 3139.350000
British Library DSC - BLDSS-3PM
British Library STI - ELD Digital store - Ingest File:
- 6346.xml