ChemInform Abstract: Diastereoselective Synthesis of 5‐Heteroaryl‐Substituted Prolines Useful for Controlling Peptide‐Bond Geometry. Issue 44 (13th October 2016)

• Record Type: Journal Article
• Authors: Ali, Rafat; Singh, Gajendra; Singh, Shalini; Ampapathi, Ravi Sankar; Haq, Wahajul
• Is Part Of: ChemInform. Volume 47:Issue 44(2016)
• Page Start: no
• Page End: no
• Publication Date: 2016-10-13
• Subjects: pyrrole derivatives -- indole derivatives, isoindole derivatives -- diastereoselective syntheses, enantioselective syntheses (incl. cis/trans‐isomerism) -- C‐C bond formation; Chemistry -- Abstracts -- Periodicals; 540.5
• DOI: 10.1002/chin.201644104
• Languages: English
• ISSNs: 0931-7597

Abstract

Abstract: A highly diastereoselective AlCl3 ‐catalyzed coupling of electron‐rich 2‐methylfuran, various indoles, and pyrrole is developed to give novel 5‐substituted L‐proline derivatives in good yields.