ChemInform Abstract: A Systematic Approach to Diverse, Lead‐Like Scaffolds from α, α‐Disubstituted Amino Acids. Issue 48 (December 2015)

• Record Type: Journal Article
• Authors: Foley, Daniel J.; Doveston, Richard G.; Churcher, Ian; Nelson, Adam; Marsden, Stephen P.
• Is Part Of: ChemInform. Volume 46:Issue 48(2015)
• Page Start: no
• Page End: no
• Publication Date: 2015-12
• Subjects: general (heterocyclic compounds) -- fused pyrimidine derivatives -- imidazole derivatives -- fused pyridine derivatives -- azepine derivatives -- oxazine derivatives -- ring closure reactions, annulation reactions; Chemistry -- Abstracts -- Periodicals; 540.5
• DOI: 10.1002/chin.201548111
• Languages: English
• ISSNs: 0931-7597

Abstract

Abstract: Four amino acid‐derived building blocks are converted into 22 scaffolds, e.g. azides (III) and (XIV), hydantoins (IV), lactams (VI), tetrahydropyridines (IX), and azepanes (XII).