2-Pyridylquinolone antimalarials with improved antimalarial activity and physicochemical properties1. Issue 7 (8th July 2015) - Charoensutthivarakul, Sitthivut
Abstract 2-Pyridylquinolones with improved solubility, an improved metabolic stability profile, reduced off-target toxicity and 12 nM Plasmodium falciparum antimalarial activity are described.