Further optimization of the mGlu5 PAM clinical candidate VU0409551/JNJ-46778212: Progress and challenges towards a back-up compound. Issue 17 (1st September 2015)

• Record Type: Journal Article
• Authors: Zhou, Ya; Malosh, Chrysa; Conde-Ceide, Susana; Martínez-Viturro, Carlos Manuel; Alcázar, Jesus; Lavreysen, Hilde; Mackie, Claire; Bridges, Thomas M.; Daniels, J. Scott; Niswender, Colleen M.; Jones, Carrie K.; Macdonald, Gregor J.; Steckler, Thomas; Conn, P. Jeffrey; Stauffer, Shaun R.; Bartolomé-Nebreda, José Manuel; Lindsley, Craig W.
• Is Part Of: Bioorganic & medicinal chemistry letters. Volume 25:Issue 17(2015)
• Page Start: 3515
• Page End: 3519
• Publication Date: 2015-09-01
• Subjects: Bioorganic chemistry -- Periodicals; Pharmaceutical chemistry -- Periodicals; 572
• DOI: 10.1016/j.bmcl.2015.06.096
• Languages: English
• ISSNs: 0960-894X

Abstract

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