Isosteric replacements of the carboxylic acid of drug candidate VX-787: Effect of charge on antiviral potency and kinase activity of azaindole-based influenza PB2 inhibitors. Issue 9 (1st May 2015)

• Record Type: Journal Article
• Authors: Boyd, Michael J.; Bandarage, Upul K.; Bennett, Hamilton; Byrn, Randal R.; Davies, Ioana; Gu, Wenxin; Jacobs, Marc; Ledeboer, Mark W.; Ledford, Brian; Leeman, Joshua R.; Perola, Emanuele; Wang, Tiansheng; Bennani, Youssef; Clark, Michael P.; Charifson, Paul S.
• Is Part Of: Bioorganic & medicinal chemistry letters. Volume 25:Issue 9(2015)
• Page Start: 1990
• Page End: 1994
• Publication Date: 2015-05-01
• Subjects: Bioorganic chemistry -- Periodicals; Pharmaceutical chemistry -- Periodicals; 572
• DOI: 10.1016/j.bmcl.2015.03.013
• Languages: English
• ISSNs: 0960-894X

Abstract

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