Regioselective sulfamoylation at low temperature enables concise syntheses of putative small molecule inhibitors of sulfatases1. Issue 18 (14th May 2015) - Miller, Duncan C.
Abstract An improved synthesis from d-glucosamine of a purported Sulf-2 inhibitor is described, with assay data for this compound and analogues showing only weak inhibition of Sulf-2, and sulfatases ARSA or ARSB.