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    Beaulieu, P. et al. (2015). Multi-parameter optimization of aza-follow-ups to BI 207524, a thumb pocket 1 HCV NS5B polymerase inhibitor. Part 2: Impact of lipophilicity on promiscuity and in vivo toxicity. Bioorganic & medicinal chemistry letters. 25 (5), pp. 1140-1145. [Online]. 
  
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