Identification of nicotinamide phosphoribosyltransferase (NAMPT) inhibitors with no evidence of CYP3A4 time-dependent inhibition and improved aqueous solubility. Issue 3 (1st February 2015)

• Record Type: Journal Article
• Authors: Zak, Mark; Liederer, Bianca M.; Sampath, Deepak; Yuen, Po-wai; Bair, Kenneth W.; Baumeister, Timm; Buckmelter, Alexandre J.; Clodfelter, Karl H.; Cheng, Eric; Crocker, Lisa; Fu, Bang; Han, Bingsong; Li, Guangkun; Ho, Yen-Ching; Lin, Jian; Liu, Xiongcai; Ly, Justin; O'Brien, Thomas; Reynolds, Dominic J.; Skelton, Nicholas; Smith, Chase C.; Tay, Suzanne; Wang, Weiru; Wang, Zhongguo; Xiao, Yang; Zhang, Lei; Zhao, Guiling; Zheng, Xiaozhang; Dragovich, Peter S.
• Is Part Of: Bioorganic & medicinal chemistry letters. Volume 25:Issue 3(2015)
• Page Start: 529
• Page End: 541
• Publication Date: 2015-02-01
• Subjects: Bioorganic chemistry -- Periodicals; Pharmaceutical chemistry -- Periodicals; 572
• DOI: 10.1016/j.bmcl.2014.12.026
• Languages: English
• ISSNs: 0960-894X

Abstract

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