Discovery of a new chemical series of BRD4(1) inhibitors using protein-ligand docking and structure-guided design. Issue 14 (15th July 2015)

• Record Type: Journal Article
• Authors: Duffy, Bryan C.; Liu, Shuang; Martin, Gregory S.; Wang, Ruifang; Hsia, Ming Min; Zhao, He; Guo, Cheng; Ellis, Michael; Quinn, John F.; Kharenko, Olesya A.; Norek, Karen; Gesner, Emily M.; Young, Peter R.; McLure, Kevin G.; Wagner, Gregory S.; Lakshminarasimhan, Damodharan; White, Andre; Suto, Robert K.; Hansen, Henrik C.; Kitchen, Douglas B.
• Is Part Of: Bioorganic & medicinal chemistry letters. Volume 25:Issue 14(2015)
• Page Start: 2818
• Page End: 2823
• Publication Date: 2015-07-15
• Subjects: Bioorganic chemistry -- Periodicals; Pharmaceutical chemistry -- Periodicals; 572
• DOI: 10.1016/j.bmcl.2015.04.107
• Languages: English
• ISSNs: 0960-894X

Abstract

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