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ISSN 2632-8682

491. Structure-based design of haloperidol analogues as inhibitors of acetyltransferase Eis from Mycobacterium tuberculosis to overcome kanamycin resistance. Issue 11 (5th October 2021)

Authors:
Punetha, Ankita; Green, Keith D.; Garzan, Atefeh; Thamban Chandrika, Nishad; Willby, Melisa J.; Pang, Allan H.; Hou, Caixia; Holbrook, Selina Y. L.; Krieger, Kyle; Posey, James E.; Parish, Tanya; Tsodikov, Oleg V.; Garneau-Tsodikova, Sylvie
Journal:
RSC medicinal chemistry
Issue:
Volume 12:Issue 11(2021)
Page Start:
1894
Record Type:
Journal Article
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493. Structure-guided discovery of selective methionyl-tRNA synthetase inhibitors with potent activity against Trypanosoma brucei. Issue 8 (18th May 2020)

Authors:
Zhang, Zhongsheng; Barros-Álvarez, Ximena; Gillespie, J. Robert; Ranade, Ranae M.; Huang, Wenlin; Shibata, Sayaka; Molasky, Nora M. R.; Faghih, Omeed; Mushtaq, Aisha; Choy, Robert K. M.; de Hostos, Eugenio; Hol, Wim G. J.; Verlinde, Christophe L. M. J.; Buckner, Frederick S.; Fan, Erkang
Journal:
RSC medicinal chemistry
Issue:
Volume 11:Issue 8(2020)
Page Start:
885
Record Type:
Journal Article
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494. Structure–activity relationship studies on 2, 5, 6-trisubstituted benzimidazoles targeting Mtb-FtsZ as antitubercular agents. Issue 1 (16th October 2020)

Authors:
Haranahalli, Krupanandan; Tong, Simon; Kim, Saerom; Awwa, Monaf; Chen, Lei; Knudson, Susan E.; Slayden, Richard A.; Singleton, Eric; Russo, Riccardo; Connell, Nancy; Ojima, Iwao
Journal:
RSC medicinal chemistry
Issue:
Volume 12:Issue 1(2021)
Page Start:
78
Record Type:
Journal Article
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495. Structure–activity relationship study of PROTACs against hematopoietic prostaglandin D2 synthase. Issue 12 (20th October 2022)

Authors:
Murakami, Yuki; Osawa, Hinata; Kurohara, Takashi; Yanase, Yuta; Ito, Takahito; Yokoo, Hidetomo; Shibata, Norihito; Naito, Mikihiko; Aritake, Kosuke; Demizu, Yosuke
Journal:
RSC medicinal chemistry
Issue:
Volume 13:Issue 12(2022)
Page Start:
1495
Record Type:
Journal Article
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497. Structure–activity relationships of valine, tert-leucine, and phenylalanine amino acid-derived synthetic cannabinoid receptor agonists related to ADB-BUTINACA, APP-BUTINACA, and ADB-P7AICA. Issue 2 (9th December 2021)

Authors:
Sparkes, Eric; Cairns, Elizabeth A.; Kevin, Richard C.; Lai, Felcia; Grafinger, Katharina Elisabeth; Chen, Shuli; Deventer, Marie H.; Ellison, Ross; Boyd, Rochelle; Martin, Lewis J.; McGregor, Iain S.; Gerona, Roy R.; Hibbs, David E.; Auwärter, Volker; Glass, Michelle; Stove, Christophe; Banister...
Journal:
RSC medicinal chemistry
Issue:
Volume 13:Issue 2(2022)
Page Start:
156
Record Type:
Journal Article
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498. Structure–property studies of an imidazoquinoline chemotype with antitrypanosomal activity. Issue 8 (10th July 2020)

Authors:
Klug, Dana M.; Diaz-Gonzalez, Rosario; DeLano, Travis J.; Mavrogiannaki, Eftychia M.; Buskes, Melissa J.; Dalton, Raeann M.; Fisher, John K.; Schneider, Katherine M.; Hilborne, Vivian; Fritsche, Melanie G.; Simpson, Quillon J.; Tear, Westley F.; Devine, William G.; Pérez-Moreno, Guiomar; Ceballos...
Journal:
RSC medicinal chemistry
Issue:
Volume 11:Issue 8(2020)
Page Start:
950
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗