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- 615.19 1
- Biochemistry -- Periodicals 1
- Bioorganic chemistry -- Periodicals 1
- Chemistry, Clinical -- Periodicals 1
- Chemistry, Organic -- Periodicals 1
- Chimie bio-organique -- Périodiques 1
- Chimie pharmaceutique -- Périodiques 1
- Nav1.7 voltage-gated sodium channel type 7 -- CIP congenital insensitivity to pain -- SCN9A sodium channel, voltage-gated, type IX, R subunit -- VGSC voltage-gated sodium channel -- SAR structure activity relationship -- hERG human Ether-à-go-go-Related Gene -- FRET Fluorescence Resonance Energy Transfer -- MIA-OA mono-iodoacetate-induced osteoarthritis -- HEK human embryonic kidney -- CNS central nervous system -- PK pharmacokinetic -- Clint, u in- vitro intrinsic clearance, unbound -- F oral bioavailability -- TFA trifluoroacetic acid -- HATU (1-[Bis(dimethylamino)methylene]-1H-1, 2, 3-triazolo[4, 5–b]pyridinium 3-oxid hexafluorophosphate) -- TBTU O-(benzotriazol-1-yl)-N, N, N′, N′-tetramethyluronium tetrafluoroborate -- DMSO dimethyl sulfoxide -- DRG Dorsal root ganglion -- LMA Locomotor assay -- SNL Spinal nerve ligation 1
- Pharmaceutical chemistry -- Periodicals 1