1. Azepino-indazoles as calcitonin gene-related peptide (CGRP) receptor antagonists. (1st January 2021) Authors: Mercer, Stephen E.; Chaturvedula, Prasad V.; Conway, Charles M.; Cook, Deborah A.; Davis, Carl D.; Pin, Sokhom S.; Macci, Robert; Schartman, Richard; Signor, Laura J.; Widmann, Kimberly A.; Whiterock, Valerie J.; Chen, Ping; Xu, Cen; Herbst, John J.; Kostich, Walter A.; Thalody, George; Macor, Jo... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 31(2021) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Calcitonin gene-related peptide (CGRP) receptor antagonists: Heterocyclic modification of a novel azepinone lead. (1st July 2021) Authors: Luo, Guanglin; Jiang, Xiang-Jun; Chen, Ling; Conway, Charles M.; Gulianello, Michael; Kostich, Walter; Keavy, Deborah; Signor, Laura J.; Chen, Ping; Davis, Carl; Whiterock, Valerie J.; Schartman, Richard; Widmann, Kimberly A.; Macor, John E.; Dubowchik, Gene M. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 43(2021) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Difluorocyclobutylacetylenes as positive allosteric modulators of mGluR5 with reduced bioactivation potential. Issue 24 (15th December 2016) Authors: Degnan, Andrew P.; Maxwell, Darrell; Balakrishnan, Anand; Brown, Jeffrey M.; Easton, Amy; Gulianello, Michael; Hanumegowda, Umesh; Hill-Drzewi, Melissa; Miller, Regina; Santone, Kenneth S.; Senapati, Arun; Shields, Eric E.; Sivarao, Digavalli V.; Westphal, Ryan; Whiterock, Valerie J.; Zhuo, Xiaol... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 24(2016) Page Start: 5871 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Oxazolidinone-based allosteric modulators of mGluR5: Defining molecular switches to create a pharmacological tool box. Issue 17 (1st September 2016) Authors: Huang, Hong; Degnan, Andrew P.; Balakrishnan, Anand; Easton, Amy; Gulianello, Michael; Huang, Yanling; Matchett, Michele; Mattson, Gail; Miller, Regina; Santone, Kenneth S.; Senapati, Arun; Shields, Eric E.; Sivarao, Digavalli V.; Snyder, Lawrence B.; Westphal, Ryan; Whiterock, Valerie J.; Yang, ... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 17(2016) Page Start: 4165 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗