1. Analysis of transition state mimicry by tight binding aminothiazoline inhibitors provides insight into catalysis by human O-GlcNAcase. Issue 6 (1st March 2016) Authors: Cekic, N.; Heinonen, J. E.; Stubbs, K. A.; Roth, C.; He, Y.; Bennet, A. J.; McEachern, E. J.; Davies, G. J.; Vocadlo, D. J. Journal: Chemical science Issue: Volume 7:Issue 6(2016:Jun.) Page Start: 3742 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Selective trihydroxylated azepane inhibitors of NagZ, a glycosidase involved in Pseudomonas aeruginosa resistance to β-lactam antibiotics. Issue 21 (17th May 2017) Authors: Bouquet, J.; King, D. T.; Vadlamani, G.; Benzie, G. R.; Iorga, B.; Ide, D.; Adachi, I.; Kato, A.; Vocadlo, D. J.; Mark, B. L.; Blériot, Y.; Désiré, J. Journal: Organic & biomolecular chemistry Issue: Volume 15:Issue 21(2017) Page Start: 4609 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Structural variation of the 3-acetamido-4, 5, 6-trihydroxyazepane iminosugar through epimerization and C-alkylation leads to low micromolar HexAB and NagZ inhibitors. Issue 3 (23rd December 2021) Authors: Bouquet, J.; Auberger, N.; Ashmus, R.; King, D.; Bordes, A.; Fontelle, N.; Nakagawa, S.; Madden, Z.; Proceviat, C.; Kato, A.; Désiré, J.; Vocadlo, D. J.; Blériot, Y. Journal: Organic & biomolecular chemistry Issue: Volume 20:Issue 3(2021) Page Start: 619 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗